EP 2988744 A4 20161102 - THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
Title (en)
THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
Title (de)
THIAZOLSUBSTITUIERTE AMINOHETEROARYLE ALS MILZTYROSINKINASEHEMMER
Title (fr)
COMPOSÉS AMINOHÉTÉROARYLE À SUBSTITUTION THIAZOLE INHIBITEURS DE TYROSINE KINASE SPLÉNIQUE
Publication
Application
Priority
- US 201361816407 P 20130426
- US 2014034909 W 20140422
Abstract (en)
[origin: WO2014176210A1] The invention provides certain thiazole-substituted aminoheteroaryl compounds of the Formula (I) or pharmaceutically acceptable salts thereof, wherein X1, X2, X3, X4, Y1, Y2, Y3, Y4, and R4 are as defined herein. The invention also provides pharmaceutical compositions comprising such compounds, and methods of using the compounds for treating diseases or conditions mediated by Spleen Tyrosine Kinase (Syk).
IPC 8 full level
A61K 31/44 (2006.01); A61K 31/426 (2006.01); A61K 31/53 (2006.01); A61P 11/00 (2006.01); A61P 19/00 (2006.01); C07D 417/12 (2006.01); C07D 417/14 (2006.01)
CPC (source: EP US)
A61K 31/4439 (2013.01 - EP US); A61K 31/497 (2013.01 - EP US); A61K 31/501 (2013.01 - EP US); A61K 31/506 (2013.01 - EP US); A61K 31/53 (2013.01 - EP US); A61P 11/00 (2017.12 - EP); A61P 19/00 (2017.12 - EP); C07D 417/12 (2013.01 - EP US); C07D 417/14 (2013.01 - EP US)
Citation (search report)
- No further relevant documents disclosed
- See references of WO 2014176210A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2014176210 A1 20141030; EP 2988744 A1 20160302; EP 2988744 A4 20161102; US 2016060255 A1 20160303; US 9745295 B2 20170829
DOCDB simple family (application)
US 2014034909 W 20140422; EP 14788026 A 20140422; US 201414786464 A 20140422