Global Patent Index - EP 3022187 A1

EP 3022187 A1 20160525 - METHOD FOR PRODUCING A 1-(5-HALONAPHTHALENE-1-SULFONYL)-1H-HEXAHYDRO-1,4-DIAZEPINE AND COMPOSITION COMPRISING SAME

Title (en)

METHOD FOR PRODUCING A 1-(5-HALONAPHTHALENE-1-SULFONYL)-1H-HEXAHYDRO-1,4-DIAZEPINE AND COMPOSITION COMPRISING SAME

Title (de)

VERFAHREN ZUR HERSTELLUNG VON 1-(5-HALONAPHTHALENE-1-SULFONYL)-1H-HEXAHYDRO-1,4-DIAZEPIN UND ZUSAMMENSETZUNG DAMIT

Title (fr)

PROCEDE POUR LA PRODUCTION D'UNE 1-(5-HALONAPHTALENE-1-SULFONYL)-1H-HEXAHYDRO-1,4-DIAZEPINE ET COMPOSITION LA COMPRENANT

Publication

EP 3022187 A1 20160525 (FR)

Application

EP 14741611 A 20140718

Priority

  • FR 1357104 A 20130718
  • EP 2014065538 W 20140718

Abstract (en)

[origin: WO2015007896A1] The invention relates to a method for the synthesis of the compounds of formula (I) wherein X is a halogen atom. The molecules ML7 (X= I) and ML9 (X= Cl) are produced by said method.

IPC 8 full level

C07D 243/08 (2006.01); A61K 31/551 (2006.01)

CPC (source: EP)

A61K 9/0048 (2013.01); A61K 47/40 (2013.01); A61P 27/02 (2017.12); C07D 243/08 (2013.01)

Citation (search report)

See references of WO 2015007896A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2015007896 A1 20150122; EP 3022187 A1 20160525; FR 3008698 A1 20150123; FR 3008698 B1 20161028; JP 2016525109 A 20160822

DOCDB simple family (application)

EP 2014065538 W 20140718; EP 14741611 A 20140718; FR 1357104 A 20130718; JP 2016526659 A 20140718