Global Patent Index - EP 3049394 A1

EP 3049394 A1 20160803 - SUBSTITUTED PHENYLALANINE DERIVATIVES AS MODULATORS OF FACTOR XIA

Title (en)

SUBSTITUTED PHENYLALANINE DERIVATIVES AS MODULATORS OF FACTOR XIA

Title (de)

SUBSTITUIERTE PHENYLALANIN-DERIVATE ALS FAKTOR XIA MODULATOREN

Title (fr)

DÉRIVÉS DE PHÉNYLALANINE SUBSTITUÉS SERVANT DE MODULATEURS DU FACTEUR XIA

Publication

EP 3049394 A1 20160803 (DE)

Application

EP 14771913 A 20140924

Priority

  • EP 13186063 A 20130926
  • EP 2014070308 W 20140924
  • EP 14771913 A 20140924

Abstract (en)

[origin: WO2015044167A1] The invention relates to substituted phenylalanine derivatives and to methods for the production thereof, in addition to the use of said derivatives for producing medicaments for the treatment and/or prophylaxis of diseases, in particular cardiovascular diseases and/or perioperative heavy blood loss.

IPC 8 full level

C07D 257/04 (2006.01); A61K 31/41 (2006.01); A61K 31/4184 (2006.01); A61K 31/4245 (2006.01); A61K 31/454 (2006.01); A61K 31/5377 (2006.01); A61P 7/00 (2006.01); A61P 9/00 (2006.01); C07D 235/26 (2006.01); C07D 271/07 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 413/12 (2006.01)

CPC (source: EP US)

A61P 7/00 (2017.12 - EP); A61P 9/00 (2017.12 - EP); C07D 231/56 (2013.01 - EP US); C07D 235/10 (2013.01 - EP US); C07D 235/26 (2013.01 - EP US); C07D 249/10 (2013.01 - EP US); C07D 249/12 (2013.01 - EP US); C07D 257/04 (2013.01 - EP US); C07D 271/07 (2013.01 - EP US); C07D 401/12 (2013.01 - EP US); C07D 401/14 (2013.01 - EP US); C07D 403/12 (2013.01 - EP US); C07D 413/12 (2013.01 - EP US)

Citation (search report)

See references of WO 2015044167A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2015044167 A1 20150402; EP 3049394 A1 20160803; US 2016244437 A1 20160825

DOCDB simple family (application)

EP 2014070308 W 20140924; EP 14771913 A 20140924; US 201415024923 A 20140924