Global Patent Index - EP 3085366 A1

EP 3085366 A1 20161026 - NMDA ANTAGONISTS FOR THE TREATMENT OF MENTAL DISORDERS WITH OCCURRENCE OF AGGRESSIVE AND/OR IMPULSIVE BEHAVIOR

Title (en)

NMDA ANTAGONISTS FOR THE TREATMENT OF MENTAL DISORDERS WITH OCCURRENCE OF AGGRESSIVE AND/OR IMPULSIVE BEHAVIOR

Title (de)

NMDA-ANTAGONISTEN ZUR BEHANDLUNG VON MENTALEN ERKRANKUNGEN MIT AUFTRETEN VON AGGRESSIVEM UND/ODER IMPULSIVEM VERHALTEN

Title (fr)

ANTAGONISTES DE NMDA POUR LE TRAITEMENT DE TROUBLES MENTAUX AVEC L'APPARITION D'UN COMPORTEMENT AGRESSIF ET/OU IMPULSIF

Publication

EP 3085366 A1 20161026 (EN)

Application

EP 15164724 A 20150422

Priority

EP 15164724 A 20150422

Abstract (en)

The present invention relates to the use of N-Methyl-D-aspartate (NMDA) antagonists at sub-anesthetic doses for the treatment of mental disorders with occurrence of aggressive and/or impulsive behavior.

IPC 8 full level

A61K 31/135 (2006.01); A61P 25/14 (2006.01)

CPC (source: EP US)

A61K 31/135 (2013.01 - EP US); A61P 25/16 (2017.12 - EP US); A61P 25/18 (2017.12 - EP US)

Citation (applicant)

  • US 5262165 A 19931116 - GOVIL SHARAD K [US], et al
  • US 5948433 A 19990907 - BURTON SCOTT ALLISON [US], et al
  • US 6010715 A 20000104 - WICK JOHN J [US], et al
  • US 6071531 A 20000606 - JONA JANAN [US], et al
  • US 3773919 A 19731120 - BOSWELL G, et al
  • MALHORTA ET AL., NEUROPSYCHOPHARMACOLOGY, vol. 17, no. 3, September 1997 (1997-09-01), pages 141 - 50
  • BREIER ET AL., AM J PSYCHIATRY, vol. 154, no. 6, June 1997 (1997-06-01), pages 805 - 11
  • COTTONE ET AL., PSYCHOPHARMACOLOGY (BERL)., vol. 226, no. 1, March 2013 (2013-03-01), pages 127 - 38
  • SCHACHT ET AL.: "Poly(ethylene glycol) Chemistry and Biological Applications", 1997, AMERICAN CHEMICAL SOCIETY, pages: 297 - 315
  • ETTMAYER ET AL., J. MED. CHEM., vol. 47, no. 10, 2004, pages 2394 - 2404
  • TESTA; MAYER: "Hydrolysis in Drug and Prodrug Metabolism: Chemistry, Biochemistry and Enzymology", 2003, WILEY-VERLAG HELVETICA CHIMICA ACTA, pages: 1 - 780
  • CONDY ET AL., BIOL PSYCHIATRY, vol. 57, 2005, pages 366 - 372

Citation (search report)

  • [XI] US 2014057988 A1 20140227 - WEG STUART [US]
  • [XI] WO 2011020061 A2 20110217 - PAPALOS DEMITRI [US]
  • [A] US 2013209585 A1 20130815 - KIM STANLEY [US]
  • [XI] DIOGO R. LARA ET AL: "Antidepressant, mood stabilizing and procognitive effects of very low dose sublingual ketamine in refractory unipolar and bipolar depression", THE INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY, vol. 16, no. 09, 20 May 2013 (2013-05-20), pages 2111 - 2117, XP055216617, ISSN: 1461-1457, DOI: 10.1017/S1461145713000485
  • [XI] BALLARD ELIZABETH D ET AL: "Improvement in suicidal ideation after ketamine infusion: Relationship to reductions in depression and anxiety", JOURNAL OF PSYCHIATRIC RESEARCH, ELSEVIER LTD, GB, vol. 58, 12 August 2014 (2014-08-12), pages 161 - 166, XP029054096, ISSN: 0022-3956, DOI: 10.1016/J.JPSYCHIRES.2014.07.027
  • [XI] MICHAEL H. BLOCH ET AL: "Effects of Ketamine in Treatment-Refractory Obsessive-Compulsive Disorder", BIOLOGICAL PSYCHIATRY, vol. 72, no. 11, 1 December 2012 (2012-12-01), pages 964 - 970, XP055216625, ISSN: 0006-3223, DOI: 10.1016/j.biopsych.2012.05.028
  • [AD] CONDY C ET AL: "Ketamine-induced distractibility: An oculomotor study in monkeys", BIOLOGICAL PSYCHIATRY, ELSEVIER SCIENCE, NEW YORK, NY; US, vol. 57, no. 4, 15 February 2005 (2005-02-15), pages 366 - 372, XP027735135, ISSN: 0006-3223, [retrieved on 20050215]
  • [A] K. SKOBLENICK ET AL: "NMDA Antagonist Ketamine Reduces Task Selectivity in Macaque Dorsolateral Prefrontal Neurons and Impairs Performance of Randomly Interleaved Prosaccades and Antisaccades", JOURNAL OF NEUROSCIENCE, vol. 32, no. 35, 29 August 2012 (2012-08-29), pages 12018 - 12027, XP055216579, ISSN: 0270-6474, DOI: 10.1523/JNEUROSCI.1510-12.2012

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

EP 3085366 A1 20161026; EP 3285752 A2 20180228; JP 2018514531 A 20180607; US 2018110742 A1 20180426; WO 2016170124 A2 20161027; WO 2016170124 A3 20170119

DOCDB simple family (application)

EP 15164724 A 20150422; EP 16721726 A 20160422; EP 2016059032 W 20160422; JP 2017555577 A 20160422; US 201715789269 A 20171020