EP 3097078 A1 20161130 - PYRIDINES AND PYRIMIDINES AND USE THEREOF
Title (en)
PYRIDINES AND PYRIMIDINES AND USE THEREOF
Title (de)
PYRIDINE UND PYRIMIDINE UND VERWENDUNG DAVON
Title (fr)
PYRIDINES ET PYRIMIDINES, ET LEUR UTILISATION
Publication
Application
Priority
- US 201461931144 P 20140124
- US 2015012591 W 20150123
Abstract (en)
[origin: WO2015112801A1] The present disclosure provides pyridines and pyrimidines of Formula I and pharmaceutically acceptable salts and solvates thereof: wherein A, G, W1, W2, W3, and R5 are defined as set forth in the specification. The present disclosure also provides uses of the compounds of Formula I and pharmaceutically acceptable salts and solvates thereof. In certain embodiments, Compounds of the present disclosure are useful for treating pain. In another embodiment, Compounds of the present disclosure are useful for treating a disorder responsive to blockade of sodium channels, or alleviating symptoms of the disorder.
IPC 8 full level
C07D 211/10 (2006.01); A61K 31/44 (2006.01); A61K 31/551 (2006.01)
CPC (source: EP US)
A61P 9/06 (2017.12 - EP); A61P 21/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/02 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 25/06 (2017.12 - EP); A61P 25/08 (2017.12 - EP); A61P 25/10 (2017.12 - EP); A61P 25/12 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 27/16 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07B 59/002 (2013.01 - US); C07D 401/04 (2013.01 - EP US); C07D 401/14 (2013.01 - EP US); C07D 403/04 (2013.01 - EP US); C07D 405/04 (2013.01 - EP US); C07D 405/14 (2013.01 - EP US); C07D 413/04 (2013.01 - EP US); C07D 413/14 (2013.01 - EP US); C07B 2200/05 (2013.01 - US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2015112801 A1 20150730; CN 106061944 A 20161026; EP 3097078 A1 20161130; EP 3097078 A4 20171129; EP 3097078 B1 20220525; JP 2017503837 A 20170202; JP 6526023 B2 20190605; US 10047075 B2 20180814; US 2017008882 A1 20170112
DOCDB simple family (application)
US 2015012591 W 20150123; CN 201580005580 A 20150123; EP 15739774 A 20150123; JP 2016548133 A 20150123; US 201515113493 A 20150123