EP 3143007 B1 20180711 - ANTIBACTERIAL QUINAZOLINE-4(3H)-ONE DERIVATIVES
Title (en)
ANTIBACTERIAL QUINAZOLINE-4(3H)-ONE DERIVATIVES
Title (de)
ANTIBAKTERIELLE CHINAZOLIN-4(3H)-ON-DERIVATE
Title (fr)
DÉRIVÉS DE QUINAZOLINE-4 ANTIBACTÉRIENNE (3H)-ONE
Publication
Application
Priority
- EP 14168718 A 20140516
- EP 2015060653 W 20150513
Abstract (en)
[origin: WO2015173329A1] The invention relates to antibacterial compounds of formula I, wherein R1 is H or halogen; R2 is the group M; R3 is H or halogen; M is MA or MB wherein A is a bond or C≡C; R1A is H or halogen; R2A is H, alkoxy or halogen; R3A is H, alkoxy, hydroxyalkoxy, hydroxyalkyl, 1,2-dihydroxyethyl, dialkylamino, 1-hydroxymethyl-cycloprop-1-yl, 1-((dimethylglycyl)oxy)methyl-cycloprop-1-yl, 3-hydroxyoxetan-3-yl, morpholin-4-ylalkyl or morpholin-4-ylalkoxy; and R1B is a group as defined in claim 1; and salts thereof.
IPC 8 full level
A61K 31/517 (2006.01); A61P 31/04 (2006.01); C07D 239/90 (2006.01)
CPC (source: CN EP KR US)
A61K 31/517 (2013.01 - EP KR US); A61P 17/00 (2017.12 - EP); A61P 31/04 (2017.12 - EP); C07D 239/90 (2013.01 - CN EP KR US); C07D 405/06 (2013.01 - EP US); Y02A 50/30 (2017.12 - EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
WO 2015173329 A1 20151119; AR 100428 A1 20161005; AU 2015261540 A1 20170112; BR 112016026787 A2 20170815; BR 112016026787 A8 20171226; CA 2948077 A1 20151119; CL 2016002918 A1 20170407; CN 106458931 A 20170222; EA 201692305 A1 20170531; EP 3143007 A1 20170322; EP 3143007 B1 20180711; ES 2687040 T3 20181023; IL 248922 A0 20170131; JP 2017515906 A 20170615; KR 20170005105 A 20170111; MX 2016014989 A 20170331; PH 12016502253 A1 20170116; SG 11201609286V A 20161229; TW 201625559 A 20160716; US 2017081292 A1 20170323; US 9796686 B2 20171024; ZA 201608680 B 20181128
DOCDB simple family (application)
EP 2015060653 W 20150513; AR P150101482 A 20150513; AU 2015261540 A 20150513; BR 112016026787 A 20150513; CA 2948077 A 20150513; CL 2016002918 A 20161116; CN 201580024307 A 20150513; EA 201692305 A 20150513; EP 15722212 A 20150513; ES 15722212 T 20150513; IL 24892216 A 20161113; JP 2017512426 A 20150513; KR 20167035088 A 20150513; MX 2016014989 A 20150513; PH 12016502253 A 20161111; SG 11201609286V A 20150513; TW 104115665 A 20150515; US 201515311758 A 20150513; ZA 201608680 A 20161215