EP 3148973 A1 20170405 - NOVEL COMPOUNDS OF THE 5-ACYLSULFANYL-HISTIDINE TYPE AS PRECURSORS OF THE CORRESPONDING 5-SULFANYLHISTIDINES AND THE DISULFIDES THEREOF
Title (en)
NOVEL COMPOUNDS OF THE 5-ACYLSULFANYL-HISTIDINE TYPE AS PRECURSORS OF THE CORRESPONDING 5-SULFANYLHISTIDINES AND THE DISULFIDES THEREOF
Title (de)
NEUARTIGE VERBINDUNGEN VOM 5-ACYLSULFANYL-HISTIDIN-TYP ALS VORLÄUFER DER ZUGEHÖRIGEN 5-SULFANYL-HISTIDINE UND DISULFIDE DAVON
Title (fr)
NOUVEAUX COMPOSES DE TYPE 5-ACYLSULFANYL-HISTIDINE EN TANT QUE PRECURSEURS DES 5-SULFANYLHISTIDINES CORRESPONDANTES ET DE LEURS DISULFURES
Publication
Application
Priority
- FR 1454935 A 20140530
- FR 2015051416 W 20150529
Abstract (en)
[origin: WO2015181507A1] The invention relates to a compound of the 5-acylsulfanyl-histidine type and the derivatives thereof, of general formula (I), wherein R1 to R3 = H, alkyl, especially CH3; R4 = H, alkyl, especially CH3, alkyle(C=0), substituted alkyl (C=O), aryl (C=O); β-alanyl (H2NCH2CH2 (C=O); α-amino-acyl; R5 = alkyl, especially methyl, phenyl. The invention also relates to the use of said compound for producing compounds of the 5-sulfanyl-histidine type and the derivatives thereof, in addition to corresponding disulfides; and to the various methods for the production thereof.
IPC 8 full level
C07D 233/84 (2006.01)
CPC (source: CN EP US)
C07D 233/84 (2013.01 - CN EP US); C07D 403/12 (2013.01 - EP US)
Citation (search report)
See references of WO 2015181507A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2015181507 A1 20151203; CA 2949334 A1 20151203; CN 106573895 A 20170419; CN 106573895 B 20201124; CN 112194632 A 20210108; EP 3148973 A1 20170405; FR 3021655 A1 20151204; FR 3021655 B1 20160708; US 2017190691 A1 20170706; US 2018258077 A1 20180913; US 9926300 B2 20180327
DOCDB simple family (application)
FR 2015051416 W 20150529; CA 2949334 A 20150529; CN 201580040441 A 20150529; CN 202010802288 A 20150529; EP 15735988 A 20150529; FR 1454935 A 20140530; US 201515314628 A 20150529; US 201815891433 A 20180208