EP 3202767 B1 20190403 - AZABICYCLO DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND MEDICAL USE THEREOF
Title (en)
AZABICYCLO DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND MEDICAL USE THEREOF
Title (de)
AZABICYCLODERIVATE, VERFAHREN ZUR HERSTELLUNG DAVON UND MEDIZINISCHE VERWENDUNG DAVON
Title (fr)
DÉRIVÉS AZABICYCLO, PROCÉDÉ DE PRÉPARATION DE CEUX-CI ET UTILISATION MÉDICALE DE CEUX-CI
Publication
Application
Priority
- CN 201410520700 A 20140930
- CN 2015090568 W 20150924
Abstract (en)
[origin: EP3202767A1] Provided are azabicyclo derivatives, a process for preparation thereof and medical use thereof. Specifically, provided are compounds of formula (I) or pharmaceutically acceptable salts, stereoisomers, solvates or prodrugs thereof, a process for preparation thereof, and application thereof in preparing EGFR (Epidermal Growth Factor Receptor) inhibitors. Definition of each group in the formula can be found in the description for details.
IPC 8 full level
C07D 487/04 (2006.01); A61K 31/53 (2006.01); A61P 35/00 (2006.01); C07D 519/00 (2006.01)
CPC (source: EP US)
A61K 31/4188 (2013.01 - EP US); A61K 31/4985 (2013.01 - EP US); A61P 35/00 (2017.12 - EP US); C07D 487/04 (2013.01 - EP US); C07D 519/00 (2013.01 - EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
EP 3202767 A1 20170809; EP 3202767 A4 20180314; EP 3202767 B1 20190403; CN 105524068 A 20160427; CN 105524068 B 20171124; JP 2017530136 A 20171012; JP 6342069 B2 20180613; US 10085983 B2 20181002; US 2017296537 A1 20171019; WO 2016050165 A1 20160407
DOCDB simple family (application)
EP 15845718 A 20150924; CN 201410520700 A 20140930; CN 2015090568 W 20150924; JP 2017517022 A 20150924; US 201515515767 A 20150924