Global Patent Index - EP 3256471 B1

EP 3256471 B1 20181212 - NOVEL 2-OXO-6,7-DIHYDROBENZO[A]QUINOLIZINE-3-CARBOXYLIC ACID DERIVATIVES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION

Title (en)

NOVEL 2-OXO-6,7-DIHYDROBENZO[A]QUINOLIZINE-3-CARBOXYLIC ACID DERIVATIVES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION

Title (de)

NEUARTIGE 2-OXO-6,7-DIHYDROBENZO[A]CHINOLIZIN-3-CARBOXYLSÄURE-DERIVATE ZUR BEHANDLUNG UND PROPHYLAXE VON HEPATITIS-B-VIRUSINFEKTION

Title (fr)

NOUVEAUX DÉRIVÉS D'ACIDE CARBOXYLIQUE 2-OXO-6,7-DIHYDROBENZO[A]QUINOLIZINE-3 POUR LE TRAITEMENT ET LA PROPHYLAXIE D'UNE INFECTION PAR LE VIRUS DE L'HÉPATITE B

Publication

EP 3256471 B1 20181212 (EN)

Application

EP 16703311 A 20160208

Priority

  • CN 2015072741 W 20150211
  • EP 2016052585 W 20160208

Abstract (en)

[origin: WO2016128335A1] The invention provides novel compounds having the general formula (I), wherein R1, R2, R3, R4, R5 and Ar are as described herein, compositions including compounds and methods of using the compounds.

IPC 8 full level

C07D 471/04 (2006.01); A61K 31/4375 (2006.01); A61P 31/12 (2006.01)

CPC (source: CN EP US)

A61P 1/16 (2017.12 - EP); A61P 31/12 (2017.12 - EP); A61P 31/20 (2017.12 - EP); C07D 471/04 (2013.01 - CN EP US)

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2016128335 A1 20160818; CN 107207505 A 20170926; CN 107207505 B 20181214; EP 3256471 A1 20171220; EP 3256471 B1 20181212; HK 1244281 B 20200207; JP 2018505198 A 20180222; JP 6435054 B2 20181205; US 10093671 B2 20181009; US 2017342069 A1 20171130

DOCDB simple family (application)

EP 2016052585 W 20160208; CN 201680008772 A 20160208; EP 16703311 A 20160208; HK 18103815 A 20180319; JP 2017542045 A 20160208; US 201715674810 A 20170811