EP 3265083 A1 20180110 - SUBSTITUTED UREA DEPSIPEPTIDE ANALOGS AS ACTIVATORS OF THE CLPP ENDOPEPTIDASE
Title (en)
SUBSTITUTED UREA DEPSIPEPTIDE ANALOGS AS ACTIVATORS OF THE CLPP ENDOPEPTIDASE
Title (de)
SUBSTITUIERTE HARNSTOFFE-DEPSIPEPTID-ANALOGA ALS AKTIVATOREN DER CLPP-ENDOPEPTIDASE
Title (fr)
ANALOGUES DE DEPSIPEPTIDE D'URÉE SUBSTITUÉS À UTILISER EN TANT QU'ACTIVATEURS DE L'ENDOPEPTIDASE CLPP
Publication
Application
Priority
- US 201562128497 P 20150304
- US 2016021043 W 20160304
Abstract (en)
[origin: WO2016141351A1] In one aspect, the invention relates to substituted urea depsipeptide analogs, derivatives thereof, and related compounds, which are useful as activators the ClpP endopeptidease; synthesis methods for making the compounds; pharmaceutical compositions comprising the compounds; and methods of treating infectious disease using the compounds and compositions. This abstract is intended as a scanning tool for purposes of searching in the particular art and is not intended to be limiting of the present invention.
IPC 8 full level
A61K 31/407 (2006.01); A61K 38/08 (2006.01); A61K 38/12 (2006.01)
CPC (source: EP US)
A61K 9/0019 (2013.01 - EP US); A61K 9/2018 (2013.01 - EP US); A61K 31/407 (2013.01 - EP US); A61K 38/12 (2013.01 - EP US); A61K 38/14 (2013.01 - EP US); A61K 38/15 (2013.01 - EP US); A61K 45/06 (2013.01 - EP US); A61K 47/02 (2013.01 - EP US); A61P 31/04 (2017.12 - EP); C07D 498/14 (2013.01 - EP US); C07D 498/22 (2013.01 - EP US); C07K 7/06 (2013.01 - EP US); C07K 11/02 (2013.01 - EP US); Y02A 50/30 (2017.12 - US)
C-Set (source: EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2016141351 A1 20160909; EP 3265083 A1 20180110; EP 3265083 A4 20181024; EP 3265083 B1 20220706; US 10100090 B2 20181016; US 10457707 B2 20191029; US 10822377 B2 20201103; US 2018079784 A1 20180322; US 2019048040 A1 20190214; US 2020031872 A1 20200130
DOCDB simple family (application)
US 2016021043 W 20160304; EP 16759625 A 20160304; US 201615554707 A 20160304; US 201816160724 A 20181015; US 201916588738 A 20190930