Global Patent Index - EP 3307749 A4

EP 3307749 A4 20190619 - HYDROPHILIC LINKERS FOR CONJUGATION

Title (en)

HYDROPHILIC LINKERS FOR CONJUGATION

Title (de)

HYDROPHILE LINKER FÜR KONJUGATION

Title (fr)

LIEURS HYDROPHILES POUR CONJUGAISON

Publication

EP 3307749 A4 20190619 (EN)

Application

EP 15773860 A 20150615

Priority

IB 2015054521 W 20150615

Abstract (en)

[origin: WO2015151078A2] Cell binding agent-drug conjugates comprising hydrophilic linkers, and methods of using such linkers and conjugates are provided.

IPC 8 full level

C07F 9/6558 (2006.01); A61K 31/537 (2006.01); A61K 38/05 (2006.01); A61K 45/06 (2006.01); A61K 47/68 (2017.01); A61P 35/00 (2006.01); C07D 207/404 (2006.01); C07D 207/46 (2006.01); C07D 213/71 (2006.01); C07D 401/12 (2006.01); C07F 9/572 (2006.01); C07F 9/58 (2006.01); C07K 5/02 (2006.01); C07K 16/32 (2006.01)

CPC (source: EP)

A61K 45/06 (2013.01); A61K 47/6803 (2017.08); A61K 47/68031 (2023.08); A61K 47/68033 (2023.08); A61K 47/68035 (2023.08); A61K 47/6855 (2017.08); A61K 47/6889 (2017.08); A61P 35/00 (2018.01); C07D 207/404 (2013.01); C07D 207/46 (2013.01); C07D 213/71 (2013.01); C07D 401/12 (2013.01); C07F 9/572 (2013.01); C07F 9/58 (2013.01); C07F 9/65583 (2013.01); C07K 5/0205 (2013.01)

Citation (search report)

  • [X] US 4003862 A 19770118 - ALBRIGHT JAMES A
  • [XDI] WO 2014080251 A1 20140530 - HANGZHOU DAC BIOTECH CO LTD [CN], et al
  • [X] FAROKH MEHRABANI ET AL: "Synthesis of new bis(tetrahydropyrrolo[3,4-b]carbazoles) with a functionalized diaryl spacer", ROYAL CHEMICAL SOCIETY. JOURNAL. PERKIN TRANSACTIONS 1, no. 12, 1 January 2001 (2001-01-01), GB, pages 1406 - 1412, XP055587069, ISSN: 1472-7781, DOI: 10.1039/b006899n
  • [X] JILA H BOAL ET AL: "Phosphorus-31 NMR studies of the kinetics of bisalkylation by isophosphoramide mustard: comparisons with phosphoramide mustard", JOURNAL OF MEDICINAL CHEMISTRY,, vol. 32, no. 8, 1 January 1989 (1989-01-01), pages 1768 - 1773, XP002453054, ISSN: 0022-2623, DOI: 10.1021/JM00128A018
  • [X] AURORE FRAIX ET AL: "Cationic lipophosphoramidates with two disulfide motifs: synthesis, behaviour in reductive media and gene transfection activity", ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 11, no. 10, 1 January 2013 (2013-01-01), pages 1650, XP055295926, ISSN: 1477-0520, DOI: 10.1039/c3ob27261c
  • [X] MYLES W. GARDNER ET AL: "Chromogenic Cross-Linker for the Characterization of Protein Structure by Infrared Multiphoton Dissociation Mass Spectrometry", ANALYTICAL CHEMISTRY, vol. 80, no. 13, 1 July 2008 (2008-07-01), US, pages 4807 - 4819, XP055587063, ISSN: 0003-2700, DOI: 10.1021/ac800625x
  • See also references of WO 2015151078A2

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2015151078 A2 20151008; WO 2015151078 A3 20160310; WO 2015151078 A4 20160714; AU 2015242210 A1 20171207; AU 2021201765 A1 20210415; AU 2021201765 B2 20221208; AU 2023200925 A1 20230323; CA 2989269 A1 20151008; CA 2989269 C 20200922; CN 108026123 A 20180511; CN 108026123 B 20210205; CN 112125929 A 20201225; EP 3307749 A2 20180418; EP 3307749 A4 20190619; NZ 737471 A 20220225

DOCDB simple family (application)

IB 2015054521 W 20150615; AU 2015242210 A 20150615; AU 2021201765 A 20210322; AU 2023200925 A 20230217; CA 2989269 A 20150615; CN 201580080839 A 20150615; CN 202011053870 A 20150615; EP 15773860 A 20150615; NZ 73747115 A 20150615