Global Patent Index - EP 3356327 A1

EP 3356327 A1 20180808 - PROCESSES FOR THE PREPARATION OF APREMILAST AND INTERMEDIATES THEREOF

Title (en)

PROCESSES FOR THE PREPARATION OF APREMILAST AND INTERMEDIATES THEREOF

Title (de)

VERFAHREN ZUR HERSTELLUNG VON APREMILAST UND ZWISCHENPRODUKTEN DAVON

Title (fr)

PROCÉDÉS DE PRÉPARATION D'APRÉMILAST, ET SES INTERMÉDIAIRES

Publication

EP 3356327 A1 20180808 (EN)

Application

EP 16778644 A 20160929

Priority

  • US 201562234094 P 20150929
  • US 2016054390 W 20160929

Abstract (en)

[origin: WO2017059040A1] Disclosed are processes for the preparation of Apremilast and intermediates for its preparation.

IPC 8 full level

C07D 209/48 (2006.01); A61K 31/4035 (2006.01); A61P 35/00 (2006.01); C07C 49/80 (2006.01); C07C 49/84 (2006.01); C07C 317/26 (2006.01)

CPC (source: EP)

A61P 35/00 (2017.12); C07C 45/63 (2013.01); C07C 49/80 (2013.01); C07C 49/84 (2013.01); C07C 317/28 (2013.01); C07C 323/22 (2013.01); C07C 323/29 (2013.01); C07C 323/41 (2013.01); C07C 323/49 (2013.01); C07D 209/48 (2013.01); C07B 2200/13 (2013.01)

Citation (search report)

See references of WO 2017059040A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2017059040 A1 20170406; EP 3356327 A1 20180808

DOCDB simple family (application)

US 2016054390 W 20160929; EP 16778644 A 20160929