EP 3383394 A1 20181010 - NOVEL ALPHA-HYDROXY CARBOXYLIC ACID AND DERIVATIVES AND OTHER GRAS- BASED PRODRUGS OF OXYMORPHONE AND USES THEREOF
Title (en)
NOVEL ALPHA-HYDROXY CARBOXYLIC ACID AND DERIVATIVES AND OTHER GRAS- BASED PRODRUGS OF OXYMORPHONE AND USES THEREOF
Title (de)
NEUARTIGE ALPHA-HYDROXY-CARBONSÄURE UND DERIVATE UND ANDERE GRAS-BASIERTE PRODRUGS VON OXYMORPHON SOWIE VERWENDUNGEN DAVON
Title (fr)
NOUVEL ACIDE ALPHA-HYDROXY CARBOXYLIQUE ET DÉRIVÉS ET AUTRES PROMÉDICAMENTS D'OXYMORPHONE À BASE DE GRAS ET LEURS UTILISATIONS
Publication
Application
Priority
- US 201514956143 A 20151201
- US 2016063836 W 20161128
Abstract (en)
[origin: US2017151228A1] The invention describes pharmaceutical compounds and compositions comprised of a ligand attached to the opioid oxymorphone, in a manner that substantially decreases or deters the potential for opioid abuse, addiction, illicit and illegal use, and overdose. When delivered at the proper dosage, the pharmaceutical composition provides therapeutic activity similar to that of the parent active agent.
IPC 8 full level
A61K 31/485 (2006.01); A61P 25/36 (2006.01); C07D 489/02 (2006.01)
CPC (source: EP US)
A61K 9/0053 (2013.01 - EP US); A61K 31/485 (2013.01 - EP US); A61K 47/542 (2017.07 - EP US); A61K 47/543 (2017.07 - US); A61P 25/36 (2017.12 - EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
US 2017151228 A1 20170601; US 2017273973 A9 20170928; US 9987269 B2 20180605; EP 3383394 A1 20181010; EP 3383394 A4 20190717; US 2018250288 A1 20180906; WO 2017095734 A1 20170608
DOCDB simple family (application)
US 201514956143 A 20151201; EP 16871311 A 20161128; US 2016063836 W 20161128; US 201815955968 A 20180418