Global Patent Index - EP 3539539 A1

EP 3539539 A1 20190918 - TABLET FORMULATIONS OF (+)-2-[1 -(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE

Title (en)

TABLET FORMULATIONS OF (+)-2-[1 -(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLINE-1,3-DIONE

Title (de)

TABLETTENFORMULIERUNGEN AUS (+)-2-[1-(3-ETHOXY-4-METHOXYPHENYL)-2-METHYLSULFONYLETHYL]-4-ACETYLAMINOISOINDOLIN-1,3-DION

Title (fr)

FORMULATIONS DE COMPRIMÉS DE (+)-2-[1+3-ETHOXY-4-MÉTHOXYPHÉNYL)-(-2-MÉTHYLSULFONYLÉTHYL]-4-ACÉTYLAMINOISOINDOLINE-1,3-DIONE

Publication

EP 3539539 A1 20190918 (EN)

Application

EP 19152029 A 20140616

Priority

  • US 201361835667 P 20130617
  • US 201361840210 P 20130627
  • EP 14735825 A 20140616
  • US 2014042456 W 20140616

Abstract (en)

Pharmaceutical compositions and single unit dosage forms of apremilast, i.e., (+)-2-[1-(3-ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione, or a pharmaceutically acceptable stereoisomer, prodrug, salt, solvate, hydrate, or clathrate, are provided herein.

IPC 8 full level

A61K 9/20 (2006.01); A61K 9/28 (2006.01); A61K 9/50 (2006.01); A61K 31/4035 (2006.01)

CPC (source: EP US)

A61K 9/2018 (2013.01 - EP US); A61K 9/2077 (2013.01 - EP US); A61K 9/2846 (2013.01 - EP US); A61K 9/2866 (2013.01 - EP US); A61K 9/5084 (2013.01 - EP US); A61K 31/4035 (2013.01 - EP US)

Citation (applicant)

  • US 201361840210 P 20130627
  • US 201361835667 P 20130617
  • US 6020358 A 20000201 - MULLER GEORGE W [US], et al
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Citation (search report)

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

US 2014370092 A1 20141218; US 9468605 B2 20161018; EP 3010490 A1 20160427; EP 3539539 A1 20190918; NZ 628329 A 20171222; WO 2014204825 A1 20141224

DOCDB simple family (application)

US 201414305082 A 20140616; EP 14735825 A 20140616; EP 19152029 A 20140616; NZ 62832914 A 20140616; US 2014042456 W 20140616