EP 3582773 A1 20191225 - PROCESSES FOR PREPARING AG-10, ITS INTERMEDIATES, AND SALTS THEREOF
Title (en)
PROCESSES FOR PREPARING AG-10, ITS INTERMEDIATES, AND SALTS THEREOF
Title (de)
VERFAHREN ZUR HERSTELLUNG VON AG-10, DESSEN ZWISCHENPRODUKTE UND SALZE DAVON
Title (fr)
PROCÉDÉS DE PRÉPARATION D'AG-10, DE SES INTERMÉDIAIRES ET DE SELS CORRESPONDANTS
Publication
Application
Priority
- US 201762460576 P 20170217
- US 2018000025 W 20180216
Abstract (en)
[origin: US2018237396A1] as well as crystalline types of Formula IX (AG-10). The processes described herein provide improved yields and efficiency, while the pharmaceutically acceptable salts and crystalline forms provide unexpected pharmacokinetic properties. Other features and aspects of the present disclosure will be apparent to a person of skill in the art upon reading the remainder of the specification.
IPC 8 full level
A61K 31/415 (2006.01); A61P 13/12 (2006.01); A61P 17/06 (2006.01)
CPC (source: CN EA EP IL KR US)
A61K 31/415 (2013.01 - CN IL); A61P 9/00 (2018.01 - CN); A61P 13/12 (2018.01 - EP); A61P 17/06 (2018.01 - EP); C07C 309/04 (2013.01 - CN EA EP KR US); C07C 309/30 (2013.01 - CN EA EP KR US); C07D 231/12 (2013.01 - CN EA EP IL KR US); A61K 31/415 (2013.01 - KR); C07B 2200/13 (2013.01 - CN EA IL KR US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
US 10513497 B2 20191224; US 2018237396 A1 20180823; AU 2018222739 A1 20190822; AU 2018222739 B2 20240314; AU 2024204057 A1 20240704; BR 112019016935 A2 20200407; CA 3051357 A1 20180823; CL 2019002321 A1 20191227; CN 110381940 A 20191025; CN 110381940 B 20230721; CN 116730920 A 20230912; CN 116730921 A 20230912; EA 201991921 A1 20200206; EP 3582773 A1 20191225; EP 3582773 A4 20210310; IL 268683 A 20191031; IL 268683 B 20221201; IL 268683 B2 20230401; IL 298196 A 20230101; JP 2020507618 A 20200312; JP 2022183220 A 20221208; JP 7157752 B2 20221020; KR 102665258 B1 20240510; KR 20190130128 A 20191121; KR 20240068787 A 20240517; MA 47511 A 20191225; MX 2019009764 A 20191111; MX 2021015220 A 20221201; MX 2022015151 A 20230201; NZ 755597 A 20230630; SG 11201906922T A 20190927; TW 201835053 A 20181001; TW 202342430 A 20231101; TW I791487 B 20230211; US 11078162 B2 20210803; US 11919865 B2 20240305; US 2020247756 A1 20200806; US 2022041558 A1 20220210; US 2024239751 A1 20240718; WO 2018151815 A1 20180823
DOCDB simple family (application)
US 201815932327 A 20180216; AU 2018222739 A 20180216; AU 2024204057 A 20240614; BR 112019016935 A 20180216; CA 3051357 A 20180216; CL 2019002321 A 20190816; CN 201880012698 A 20180216; CN 202310822637 A 20180216; CN 202310822802 A 20180216; EA 201991921 A 20180216; EP 18753963 A 20180216; IL 26868319 A 20190813; IL 29819622 A 20221114; JP 2019545281 A 20180216; JP 2022162530 A 20221007; KR 20197026567 A 20180216; KR 20247015025 A 20180216; MA 47511 A 20180216; MX 2019009764 A 20180216; MX 2021015220 A 20180216; MX 2022015151 A 20190815; NZ 75559718 A 20180216; SG 11201906922T A 20180216; TW 107105862 A 20180221; TW 112100724 A 20180221; US 2018000025 W 20180216; US 201916676931 A 20191107; US 202117350066 A 20210617; US 202418413175 A 20240116