EP 3645534 A1 20200506 - REINFORCED MACROCYCLIC LIGANDS, COMPLEXES THEREOF, AND USES OF SAME
Title (en)
REINFORCED MACROCYCLIC LIGANDS, COMPLEXES THEREOF, AND USES OF SAME
Title (de)
VERSTÄRKTE MAKROCYCLISCHE LIGANDEN, KOMPLEXE DAVON UND VERWENDUNGEN DAVON
Title (fr)
LIGANDS MACROCYCLIQUES RENFORCÉS, LEURS COMPLEXES AINSI QUE LEURS UTILISATIONS
Publication
Application
Priority
- FR 1755933 A 20170628
- EP 2018067482 W 20180628
Abstract (en)
[origin: WO2019002505A1] The invention relates to new macrocyclic ligands of formula (I) and complexes thereof, particularly radioactive complexes, and to the uses thereof and a method for preparing same. The ligands have a reinforced pyclene core.
IPC 8 full level
A61K 31/439 (2006.01); A61P 35/00 (2006.01); C07D 471/18 (2006.01)
CPC (source: EP US)
C07D 471/18 (2013.01 - EP US); A61K 9/0019 (2013.01 - US); A61K 51/0482 (2013.01 - US); A61K 51/121 (2013.01 - US)
Citation (search report)
See references of WO 2019002505A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2019002505 A1 20190103; EP 3645534 A1 20200506; FR 3068355 A1 20190104; FR 3068355 B1 20201211; US 11155553 B2 20211026; US 2020157101 A1 20200521
DOCDB simple family (application)
EP 2018067482 W 20180628; EP 18733626 A 20180628; FR 1755933 A 20170628; US 201816626645 A 20180628