Global Patent Index - EP 3656391 A1

EP 3656391 A1 20200527 - IMMUNE SYSTEM MODULATORS

Title (en)

IMMUNE SYSTEM MODULATORS

Title (de)

IMMUNSYSTEMMODULATOREN

Title (fr)

MODULATEURS DU SYSTÈME IMMUNITAIRE

Publication

EP 3656391 A1 20200527 (EN)

Application

EP 19204654 A 20140908

Priority

  • US 201361875598 P 20130909
  • EP 14771713 A 20140908
  • US 2014054612 W 20140908

Abstract (en)

The present invention described herein relates to compositions that interact with molecules that suppress the immune system. More specifically, embodiments described herein concern the discovery, manufacture, and use of compositions that remove immunosuppression the immune system by binding to immunoregulatory peptides that interact with receptors on immune cells, compositions the can stimulate immune cells, and compositions that are cytotoxic to tumor cells.

IPC 8 full level

A61K 38/00 (2006.01); C07K 7/06 (2006.01); C07K 7/08 (2006.01); C07K 14/705 (2006.01); C07K 14/715 (2006.01); G01N 33/566 (2006.01)

CPC (source: EP US)

A61P 35/00 (2017.12 - EP); C07K 7/06 (2013.01 - US); C07K 7/08 (2013.01 - US); C07K 14/70546 (2013.01 - EP US); C07K 14/7155 (2013.01 - EP US); C07K 14/76 (2013.01 - EP US); A61K 38/00 (2013.01 - EP US); C07K 2319/00 (2013.01 - US)

Citation (applicant)

  • US 7960126 B2 20110614 - HAAKANSSON LEIF [SE], et al
  • US 8110347 B2 20120207 - HAAKANSSON LEIF [SE], et al
  • US 2010323370 A1 20101223 - HAKANSSON LEIF [SE], et al
  • US 2011262470 A1 20111027 - HAKANSSON LEIF [SE], et al
  • US 8142784 B2 20120327 - EBENS JR ALLEN J [US], et al
  • US 7628986 B2 20091208 - WEBER RICHARD [US], et al
  • US 5591669 A 19970107 - KRIMPENFORT PAULUS J A [NL], et al
  • US 5589369 A 19961231 - SEIDMAN JONATHAN G [US], et al
  • US 5545807 A 19960813 - SURANI AZIM M [GB], et al
  • US 5565332 A 19961015 - HOOGENBOOM HENDRICUS R J M [GB], et al
  • US 5573905 A 19961112 - LERNER RICHARD [US], et al
  • US 7985840 B2 20110726 - FUH GERMAINE [US], et al
  • US 5567610 A 19961022 - BORREBAECK CARL [SE], et al
  • US 5229275 A 19930720 - GOROFF DIANA K [US]
  • US 6495674 B1 20021217 - LEMKE GREG ERWIN [US], et al
  • US 4215051 A 19800729 - PALMER DAIVD A [US], et al
  • US 8153758 B2 20120410 - MIAO ZHENWEI [US], et al
  • US 7888533 B2 20110215 - TIAN FENG [US], et al
  • US 6344483 B1 20020205 - HALLINAN E ANN [US], et al
  • US 7957912 B2 20110607 - SELIFONOV SERGEY A [US], et al
  • US 6881719 B2 20050419 - SARAGOVI HORACIO URI [CA], et al
  • US 7816324 B2 20101019 - AHN JUNG-MO [US], et al
  • US 7153685 B2 20061226 - MAO CHENGJIAN [US], et al
  • US 7589170 B1 20090915 - SMYTHE MARK LESLIE [AU], et al
  • US 7252952 B2 20070807 - LORENS JAMES B [NO], et al
  • WO 9509344 A1 19950406 - DATALINER AB [SE], et al
  • US 7745607 B2 20100629 - LI YINGFU [CA], et al
  • WO 0193911 A2 20011213 - TRUSTESS OF THE UNIVERSITY OF [US]
  • WO 03000778 A1 20030103 - SAMYANG CORP [KR]
  • EP 0681481 A1 19951115 - CHIESI FARMA SPA [IT]
  • WO 2004064731 A2 20040805 - UNIV WASHINGTON [US]
  • US 7736653 B2 20100615 - KIM YOUNG MIN [KR], et al
  • US 8133688 B2 20120313 - HAKANSSON LEIF [SE], et al
  • US 7572906 B2 20090811 - DROPULIC BORO [US], et al
  • US 8012468 B2 20110906 - KIM TAI-GYU [KR], et al
  • US 8182983 B2 20120522 - HAKANSSON LEIF [SE], et al
  • DUNN GP ET AL., IMMUNITY, vol. 21, 2004, pages 137 - 148
  • SCHULE J ET AL., BREAST CANCER RES TREAT., vol. 74, 2002, pages 33 - 40
  • WOLFRAM RM ET AL., INT J CANCER., vol. 88, 2000, pages 239 - 44
  • PETERSEN RP ET AL., CANCER, vol. 107, 2006, pages 2866 - 72
  • CLINCHY B ET AL., CANCER, vol. 109, 2007, pages 1742 - 9
  • GALON J ET AL., SCIENCE, vol. 313, 2006, pages 1960 - 4
  • MLECNIK B ET AL., J CLIN ONCOL, vol. 29, 2011, pages 610 - 8
  • GORELIK E. ET AL., ADV CANCER RES., vol. 39, 1983, pages 71 - 120
  • VOSE BM ET AL., INT J CANCER, vol. 20, 1977, pages 895 - 902
  • MENETRIER-CAUX C ET AL., BR J CANCER, vol. 79, 1999, pages 119 - 130
  • HEIMDAL JH ET AL., SCAND J IMMUNOL, vol. 51, 2000, pages 271 - 278
  • HEIMDAL JH ET AL., SCAND J IMMUNOL, vol. 53, 2001, pages 162 - 170
  • KIM R ET AL., CANCER RES., vol. 66, no. 11, 1 June 2006 (2006-06-01), pages 5527 - 36
  • MOCELLIN S ET AL., J IMMUNOTHER, vol. 24, 2001, pages 392 - 407
  • PERDRIZET GA ET AL., J EXP MED., vol. 171, 1990, pages 1205 - 20
  • YU P ET AL., J EXP MED., vol. 201, 2005, pages 779 - 91
  • KOEBEL CM ET AL., NATURE, vol. 450, 2007, pages 903 - 7
  • TENG MW ET AL., J LEUKOC BIOL., vol. 84, 2008, pages 988 - 93
  • GAJEWSKI TF ET AL., J IMMUNOTHER, vol. 29, 2006, pages 233 - 40
  • WHITESIDE TL, ONCOGENE, vol. 27, 2008, pages 5904 - 12
  • WANEBO HJ ET AL., CANCER, vol. 57, 1986, pages 656 - 62
  • MANTOVANI, G. ET AL., DIAGN. CLIN. IMMUNOL., vol. 5, 1987, pages 104 - 111
  • LAUEROVA L ET AL., NEOPLASMA, vol. 46, 1999, pages 141 - 149
  • TSUBONO M ET AL., J CLIN LAB IMMUNOL, vol. 33, 1990, pages 107 - 115
  • PELLEGRINI P ET AL., CANCER IMMUNOL IMMUNOTHER, vol. 42, 1996, pages 1 - 8
  • BOTTI C ET AL., INTL J BIOL MARKERS, vol. 13, 1998, pages 51 - 69
  • HOGG N ET AL., J CELL SCI., vol. 116, 2003, pages 4695 - 705
  • GIBLIN PA ET AL., CURR PHARM DES., vol. 12, 2006, pages 2771 - 95
  • EVANS R ET AL., CELL SCI., vol. 122, 2009, pages 215 - 25
  • VYTH-DREESE FA, EUR J IMMUNOL., vol. 12, 1993, pages 3292 - 9
  • CULP WD ET AL., J PROTEOMERES, vol. 5, 2006, pages 1332 - 43
  • VYTH-DREESE ET AL., EUR. J. IMMUNOL., vol. 12, 1993, pages 3292 - 3299
  • CHOTHIALESK, J. MOL. BIOL., vol. 196, 1987, pages 901 - 917
  • CHOTHIA ET AL., NATURE, vol. 342, 1989, pages 878 - 883
  • JAKOBOVITS ET AL., PROC. NATL. ACAD. SCI. USA, vol. 90, 1993, pages 2551
  • JAKOBOVITS ET AL., NATURE, vol. 362, 1993, pages 255 - 258
  • BRUGGERMANN ET AL., YEAR IN IMMUNO, vol. 7, 1993, pages 33
  • MCCAFFERTY ET AL., NATURE, vol. 348, 1990, pages 552 - 553
  • JOHNSON, KEVIN S.CHISWELL, DAVID J., CURRENT OPINION IN STRUCTURAL BIOLOGY, vol. 3, 1993, pages 564 - 571
  • MARKS ET AL., J. MOL. BIOL., vol. 222, 1991, pages 581 - 597
  • GRIFFITH ET AL., EMBO J., vol. 12, 1993, pages 725 - 734
  • LOGANSHENK, PROC. NATL. ACAD. SCI. USA, vol. 81, 1984, pages 3655 - 3659
  • RUTHER ET AL., EMBO J., vol. 2, 1983, pages 1791
  • INOUYEINOUYE, NUCLEIC ACIDS RES., vol. 13, 1985, pages 3101 - 3109
  • VAN HEEKESCHUSTER, J. BIOL. CHEM., vol. 264, 1989, pages 5503 - 5509
  • SMITH ET AL., J. VIROL., vol. 46, 1983, pages 584
  • QU, ALEAHY, DJ, PROC. NATL. ACAD. SCI. USA, vol. 92, 1995, pages 10277 - 10281
  • MALAKAUSKASMAYO: "Design, Structure and Stability of a Hyperthermophilic Protein Variant", NATURE STRUC. BIOL., vol. 5, 1998, pages 470, XP008008261, DOI: 10.1038/nsb0698-470
  • DAHIYATMAYO: "De Novo Protein Design: Fully Automated Sequence Selection", SCIENCE, vol. 278, 1997, pages 82 - 87
  • DEGRADO: "Proteins from Scratch", SCIENCE, vol. 278, 1997, pages 80 - 81
  • DAHIYATSARISKYMAYO: "De Novo Protein Design: Towards Fully Automated Sequence Selection", J. MOL. BIOL., vol. 273, 1997, pages 789 - 796
  • DAHIYATMAYO: "Probing the Role of Pachng Specificity in Protein Design", PROC. NATL. ACAD. SCI. USA, vol. 94, 1997, pages 10172 - 10177
  • HELLINGA: "Rational Protein Design--Combining Theory and Experiment", PROC. NATL. ACAD. SCI. USA, vol. 94, 1997, pages 10015 - 10017
  • SUMAYO: "Coupling Backbone Flexibility and Amino Acid Sequence Selection in Protein Design", PROT. SCI., vol. 6, 1997, pages 1701 - 1707
  • DAHIYATGORDONMAYO: "Automated Design of the Surface Positions of Protein Helices", PROT. SCI., vol. 6, 1997, pages 1333 - 1337, XP000982615
  • DAHIYATMAYO: "Protein Design Automation", PROT. SCI., vol. 5, 1996, pages 895 - 903, XP002073372
  • CHEN ET AL., ACS CHEMICAL BIOLOGY, vol. 4, no. 9, 2009, pages 769 - 81
  • BIOCHEM. BIOPHYS. RES. COMMUN., vol. 102, 1981, pages 1048 - 1054
  • J. NATL. CANC. INST., vol. 80, 1988, pages 1154 - 1159
  • CANCER RES., vol. 48, 1988, pages 6097 - 6102
  • PROC. NATL. ACAD. SCI., vol. 79, 1982, pages 626 - 629
  • "Remington's Pharmaceutical Sciences", 1990, MACK PUBLISHING COMPANY
  • "handbook of Pharmaceutical Excipients", 2000, PHARMACEUTICAL PRESS
  • WANG ET AL., SCIENCE, vol. 310, no. 5751, 2005, pages 1159 - 1163
  • STAUBER ET AL., PROC. NATL. ACAD. SCI. USA, vol. 103, no. 8, 2006, pages 2788 - 2793
  • MA Q ET AL., J BIOL CHEM., vol. 277, 2002, pages 10638 - 41
  • "UniProt", Database accession no. P20701

Citation (search report)

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2015035332 A1 20150312; AU 2014317884 B2 20170907; CA 2923160 A1 20150312; CN 105744944 A 20160706; CN 105744944 B 20200707; CN 111732652 A 20201002; DK 3043810 T3 20200127; EP 3043810 A1 20160720; EP 3043810 B1 20191023; EP 3656391 A1 20200527; ES 2777939 T3 20200806; JP 2016531583 A 20161013; JP 2020019803 A 20200206; JP 6886816 B2 20210616; KR 102162323 B1 20201006; KR 20160054531 A 20160516; US 10301356 B2 20190528; US 2016311854 A1 20161027; US 2017298096 A1 20171019; US 2019375789 A1 20191212; US 9657059 B2 20170523

DOCDB simple family (application)

US 2014054612 W 20140908; AU 2014317884 A 20140908; CA 2923160 A 20140908; CN 201480061392 A 20140908; CN 202010645072 A 20140908; DK 14771713 T 20140908; EP 14771713 A 20140908; EP 19204654 A 20140908; ES 14771713 T 20140908; JP 2016540471 A 20140908; JP 2019183568 A 20191004; KR 20167008914 A 20140908; US 201414916512 A 20140908; US 201715488283 A 20170414; US 201916379654 A 20190409