Global Patent Index - EP 3665169 A1

EP 3665169 A1 20200617 - CARBOXAMIDES AS UBIQUITIN-SPECIFIC PROTEASE INHIBITORS

Title (en)

CARBOXAMIDES AS UBIQUITIN-SPECIFIC PROTEASE INHIBITORS

Title (de)

CARBOXAMIDE ALS UBIQUITIN-SPEZIFISCHE PROTEASEINHIBITOREN

Title (fr)

CARBOXAMIDES UTILISÉES EN TANT QU'INHIBITEURS DE PROTÉASE SPÉCIFIQUE DE L'UBIQUITINE

Publication

EP 3665169 A1 20200617 (EN)

Application

EP 18760137 A 20180809

Priority

  • US 201762544083 P 20170811
  • US 2018046061 W 20180809

Abstract (en)

[origin: WO2019032863A1] The present disclosure relates to modulators, such as inhibitors, of at least one pathway chosen from USP28 and USP25, pharmaceutical compositions comprising the inhibitors, and methods of using the inhibitors. The modulators, such as inhibitors, of at least one pathway chosen from USP28 and USP25 can be useful in the treatment of cancers, among other ailments.

IPC 8 full level

C07D 405/14 (2006.01); A61K 31/4365 (2006.01); A61K 31/496 (2006.01); A61K 31/4995 (2006.01); A61K 31/5386 (2006.01); A61K 31/551 (2006.01); A61P 35/00 (2006.01); C07D 471/04 (2006.01); C07D 487/04 (2006.01); C07D 495/04 (2006.01); C07D 519/00 (2006.01)

CPC (source: EP US)

A61P 35/00 (2017.12 - EP); C07D 405/14 (2013.01 - EP); C07D 471/04 (2013.01 - EP); C07D 487/04 (2013.01 - EP); C07D 495/04 (2013.01 - EP US); C07D 519/00 (2013.01 - EP US)

Citation (search report)

See references of WO 2019032863A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2019032863 A1 20190214; AR 112468 A1 20191030; AU 2018316254 A1 20200220; AU 2018316254 B2 20220714; CA 3072449 A1 20190214; EP 3665169 A1 20200617; JP 2020530469 A 20201022; MA 49841 A 20200617; TW 201920157 A 20190601; US 11524966 B1 20221213

DOCDB simple family (application)

US 2018046061 W 20180809; AR P180102268 A 20180809; AU 2018316254 A 20180809; CA 3072449 A 20180809; EP 18760137 A 20180809; JP 2020507569 A 20180809; MA 49841 A 20180809; TW 107127893 A 20180809; US 201816637692 A 20180809