Global Patent Index - EP 3681485 A1

EP 3681485 A1 20200722 - PHARMACEUTICAL COMPOSITION

Title (en)

PHARMACEUTICAL COMPOSITION

Title (de)

PHARMAZEUTISCHE ZUSAMMENSETZUNG

Title (fr)

COMPOSITION PHARMACEUTIQUE

Publication

EP 3681485 A1 20200722 (EN)

Application

EP 18779051 A 20180911

Priority

  • US 201762557298 P 20170912
  • IB 2018056904 W 20180911

Abstract (en)

[origin: US2019076418A1] The present invention relates to a pharmaceutical composition for oral administration comprising a non-bile farnesoid X receptor (FXR) agonist 2-[(1R,3R,5S)-3-({5-cyclopropyl-3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-4-yl}methoxy)-8-azabicyclo[3.2.1]octan-8-yl]-4-fluoro-1,3-benzothiazole-6-carboxylic acid, or a pharmaceutically acceptable salt thereof, and at least one lipid excipient; to a capsule for oral administration comprising said pharmaceutical composition; to the use of said pharmaceutical composition for the treatment of a FXR mediated disorder or condition; and to a process for preparing said pharmaceutical composition.

IPC 8 full level

A61K 9/48 (2006.01); A61K 9/08 (2006.01); A61K 47/14 (2017.01)

CPC (source: EP KR US)

A61K 9/0095 (2013.01 - KR); A61K 9/08 (2013.01 - EP KR US); A61K 9/4825 (2013.01 - US); A61K 9/4858 (2013.01 - EP KR US); A61K 9/4866 (2013.01 - US); A61K 31/46 (2013.01 - EP KR US); A61K 47/14 (2013.01 - EP KR US); A61P 1/16 (2017.12 - EP KR US); A61K 9/4833 (2013.01 - US)

Citation (search report)

See references of WO 2019053581A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

US 11207313 B2 20211228; US 2019076418 A1 20190314; AR 114930 A1 20201111; AU 2018332191 A1 20200220; AU 2018332191 B2 20210520; BR 112020004663 A2 20200915; CA 3072559 A1 20190321; CL 2020000601 A1 20200911; CN 111093637 A 20200501; EP 3681485 A1 20200722; IL 272419 A 20200331; JP 2020533297 A 20201119; KR 20200052280 A 20200514; MX 2020002432 A 20200713; RU 2020111980 A 20211013; RU 2020111980 A3 20211123; TW 201919626 A 20190601; US 2022071983 A1 20220310; WO 2019053581 A1 20190321

DOCDB simple family (application)

US 201816125809 A 20180910; AR P180102544 A 20180907; AU 2018332191 A 20180911; BR 112020004663 A 20180911; CA 3072559 A 20180911; CL 2020000601 A 20200310; CN 201880057264 A 20180911; EP 18779051 A 20180911; IB 2018056904 W 20180911; IL 27241920 A 20200202; JP 2020513606 A 20180911; KR 20207006661 A 20180911; MX 2020002432 A 20180911; RU 2020111980 A 20180911; TW 107131663 A 20180910; US 202117529078 A 20211117