Global Patent Index - EP 3704126 A4

EP 3704126 A4 20201209 - COMPOUNDS AND USE THEREOF IN THE EXPANSION OF STEM CELLS AND/OR PROGENITOR CELLS

Title (en)

COMPOUNDS AND USE THEREOF IN THE EXPANSION OF STEM CELLS AND/OR PROGENITOR CELLS

Title (de)

VERBINDUNGEN UND VERWENDUNG DAVON IN DER EXPANSION VON STAMMZELLEN UND/ODER VORLÄUFERZELLEN

Title (fr)

COMPOSÉS ET LEUR UTILISATION DANS L'EXPANSION DE CELLULES SOUCHES ET/OU DE CELLULES PROGÉNITRICES

Publication

EP 3704126 A4 20201209 (EN)

Application

EP 18872845 A 20181101

Priority

  • US 201762581149 P 20171103
  • IB 2018058593 W 20181101

Abstract (en)

[origin: WO2019087129A1] The invention relates to compounds of formula I and pharmaceutical compositions containing them. Also, the invention relates to methods for expanding stem cells and/or progenitor cells and methods for treating a hematopoietic disorder/malignancy, and autoimmune disease and/or an inherited immunodeficient disease (I).

IPC 8 full level

C07D 495/04 (2006.01); A61K 31/343 (2006.01); A61K 31/381 (2006.01); A61K 31/4355 (2006.01); A61K 31/4365 (2006.01); A61K 31/444 (2006.01); A61K 31/4709 (2006.01); A61K 31/4725 (2006.01); A61K 31/501 (2006.01); A61K 31/506 (2006.01); A61P 35/02 (2006.01); A61P 37/02 (2006.01); A61P 43/00 (2006.01); C07D 333/70 (2006.01); C07D 491/048 (2006.01); C12N 5/02 (2006.01); C12N 5/071 (2010.01); C12N 5/0789 (2010.01)

CPC (source: EP IL KR US)

A61K 31/343 (2013.01 - EP IL); A61K 31/381 (2013.01 - EP IL KR); A61K 31/4355 (2013.01 - EP IL KR); A61K 31/4365 (2013.01 - EP IL KR); A61K 31/444 (2013.01 - EP IL); A61K 31/4709 (2013.01 - EP IL); A61K 31/4725 (2013.01 - EP IL); A61K 31/501 (2013.01 - EP IL); A61K 31/506 (2013.01 - EP IL); A61K 31/519 (2013.01 - EP IL); A61K 35/28 (2013.01 - EP IL KR US); A61P 35/00 (2018.01 - IL KR); A61P 37/00 (2018.01 - IL KR); C07D 333/66 (2013.01 - IL US); C07D 333/70 (2013.01 - EP IL KR US); C07D 409/12 (2013.01 - US); C07D 491/04 (2013.01 - IL KR); C07D 491/048 (2013.01 - EP IL); C07D 495/04 (2013.01 - EP IL KR US); C12N 5/0607 (2013.01 - IL US); C12N 5/0647 (2013.01 - EP IL KR); A61K 2300/00 (2013.01 - IL KR); C12N 2500/30 (2013.01 - IL US); C12N 2501/999 (2013.01 - EP IL KR)

C-Set (source: EP)

  1. A61K 31/519 + A61K 2300/00
  2. A61K 31/381 + A61K 2300/00
  3. A61K 31/4355 + A61K 2300/00
  4. A61K 31/4365 + A61K 2300/00

Citation (search report)

  • [Y] WO 2011147764 A1 20111201 - ORGANON NV [NL], et al
  • [Y] WO 2013126856 A1 20130829 - UNIV VANDERBILT [US]
  • [Y] WO 2004058747 A1 20040715 - ARTHRON LTD [AU], et al
  • [Y] WO 9822452 A1 19980528 - KYOWA HAKKO KOGYO KK [JP], et al
  • [X] PABST CAROLINE ET AL: "A High-Throughput Screen to Identify Compounds Preserving Primary Human AML Stem Cells Ex-Vivo", BLOOD, vol. 118, no. 21, November 2011 (2011-11-01), & 53RD ANNUAL MEETING AND EXPOSITION OF THE AMERICAN-SOCIETY-OF-HEMATOLOGY (ASH); SAN DIEGO, CA, USA; DECEMBER 10 -13, 2011, pages 1531, XP002800869
  • [X] FARES IMAN HATEM ET AL: "Screen for Small Molecules Capable of Expanding Human Hematopoietic Stem Cell Ex Vivo", BLOOD, vol. 118, no. 21, November 2011 (2011-11-01), & 53RD ANNUAL MEETING AND EXPOSITION OF THE AMERICAN-SOCIETY-OF-HEMATOLOGY (ASH); SAN DIEGO, CA, USA; DECEMBER 10 -13, 2011, pages 836 - 837, XP002800870
  • [X] SZTUBA-SOLINSKA J ET AL: "Identification of biologically active, HIV TAR RNA-binding small molecules using small molecule microarrays", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 20140611 AMERICAN CHEMICAL SOCIETY USA, vol. 136, no. 23, 11 June 2014 (2014-06-11), pages 8402 - 8410, XP002800871, DOI: 10.1021/JA502754F
  • See also references of WO 2019087129A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2019087129 A1 20190509; AU 2018361971 A1 20200604; AU 2023241382 A1 20231026; BR 112020008330 A2 20201006; CA 3080695 A1 20190509; CN 111417640 A 20200714; CN 111417640 B 20240405; EP 3704126 A1 20200909; EP 3704126 A4 20201209; IL 274291 A 20200630; IL 274291 B1 20230601; IL 274291 B2 20231001; JP 2021501582 A 20210121; KR 20200084873 A 20200713; MX 2020004414 A 20201019; SG 11202003807R A 20200528; US 11696928 B2 20230711; US 2020323923 A1 20201015; US 2023338429 A1 20231026

DOCDB simple family (application)

IB 2018058593 W 20181101; AU 2018361971 A 20181101; AU 2023241382 A 20231006; BR 112020008330 A 20181101; CA 3080695 A 20181101; CN 201880074165 A 20181101; EP 18872845 A 20181101; IL 27429120 A 20200427; JP 2020524269 A 20181101; KR 20207015361 A 20181101; MX 2020004414 A 20181101; SG 11202003807R A 20181101; US 201816760780 A 20181101; US 202318320929 A 20230519