EP 3805231 A1 20210414 - INHIBITOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF
Title (en)
INHIBITOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF
Title (de)
INHIBITORHALTIGES TRICYCLISCHES DERIVAT, HERSTELLUNGSVERFAHREN DAFÜR UND VERWENDUNG DAVON
Title (fr)
INHIBITEUR CONTENANT UN DÉRIVÉ TRICYCLIQUE, SON PROCÉDÉ DE PRÉPARATION ET SON APPLICATION
Publication
Application
Priority
- CN 201810541998 A 20180530
- CN 201810772171 A 20180713
- CN 201811142142 A 20180928
- CN 201910176302 A 20190308
- CN 2019088788 W 20190528
Abstract (en)
An inhibitor containing a tricyclic derivative, a preparation method therefor and a pharmaceutical composition comprising the inhibitor, as well as a use thereof as a phosphoinositide 3 kinase (PI3K) inhibitor in the treatment of cancer and diseases or conditions mediated by or dependent on PI3K imbalance.
IPC 8 full level
C07D 498/04 (2006.01); A61K 31/4162 (2006.01); A61K 31/4188 (2006.01); A61K 31/4196 (2006.01); A61K 31/553 (2006.01); A61P 35/00 (2006.01); C07D 498/14 (2006.01)
CPC (source: CN EP KR US)
A61K 31/4188 (2013.01 - KR); A61K 31/422 (2013.01 - KR); A61K 31/553 (2013.01 - KR); A61P 3/00 (2018.01 - CN); A61P 9/00 (2018.01 - CN); A61P 11/00 (2018.01 - CN); A61P 19/00 (2018.01 - CN); A61P 25/00 (2018.01 - CN); A61P 29/00 (2018.01 - CN); A61P 35/00 (2018.01 - CN EP KR US); A61P 35/02 (2018.01 - CN); A61P 37/02 (2018.01 - CN); C07D 498/04 (2013.01 - CN EP KR US); C07D 498/10 (2013.01 - CN); C07D 498/14 (2013.01 - CN EP KR US); C07D 519/00 (2013.01 - CN EP)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
EP 3805231 A1 20210414; EP 3805231 A4 20220112; AU 2019276514 A1 20201126; AU 2019276514 B2 20231214; BR 112020022328 A2 20210202; CA 3101227 A1 20191205; CN 110785423 A 20200211; CN 110785423 B 20220726; CN 114835729 A 20220802; CN 114835729 B 20240531; JP 2021525252 A 20210924; JP 2024083359 A 20240621; JP 7456945 B2 20240327; KR 20210018304 A 20210217; MX 2020012347 A 20210129; TW 202016120 A 20200501; US 2021221822 A1 20210722; WO 2019228341 A1 20191205
DOCDB simple family (application)
EP 19810781 A 20190528; AU 2019276514 A 20190528; BR 112020022328 A 20190528; CA 3101227 A 20190528; CN 2019088788 W 20190528; CN 201980002845 A 20190528; CN 202210657073 A 20190528; JP 2020565398 A 20190528; JP 2024040496 A 20240314; KR 20207036502 A 20190528; MX 2020012347 A 20190528; TW 108118756 A 20190530; US 201917059936 A 20190528