Global Patent Index - EP 3810623 A1

EP 3810623 A1 20210428 - A NOVEL PROCESS FOR THE PREPARATION OF SGLT-2 INHIBITORS

Title (en)

A NOVEL PROCESS FOR THE PREPARATION OF SGLT-2 INHIBITORS

Title (de)

NEUES VERFAHREN ZUR HERSTELLUNG VON SGLT-2-INHIBITOREN

Title (fr)

NOUVEAU PROCÉDÉ DE PRÉPARATION D'INHIBITEURS DE SGLT-2

Publication

EP 3810623 A1 20210428 (EN)

Application

EP 19742290 A 20190621

Priority

  • EP 2018025170 W 20180625
  • EP 2019025192 W 20190621

Abstract (en)

[origin: WO2020001812A1] The present invention relates to a novel process for the preparation of SGLT-2 inhibitors via addition of a hydroxymethylene group in an open chain intermediate, readily accessible from D-glucose.

IPC 8 full level

C07C 43/18 (2006.01); C07F 7/18 (2006.01); C07H 7/04 (2006.01); C07H 9/04 (2006.01); C07H 23/00 (2006.01)

CPC (source: EP)

C07F 7/1804 (2013.01); C07H 1/00 (2013.01); C07H 7/04 (2013.01); C07H 9/04 (2013.01); C07H 23/00 (2013.01)

Citation (search report)

See references of WO 2020001812A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2020001812 A1 20200102; EP 3810623 A1 20210428

DOCDB simple family (application)

EP 2019025192 W 20190621; EP 19742290 A 20190621