EP 3823617 B1 20240306 - ENANTIOMERICALLY PURIFIED GPER AGONIST FOR USE IN TREATING DISEASE STATES AND CONDITIONS
Title (en)
ENANTIOMERICALLY PURIFIED GPER AGONIST FOR USE IN TREATING DISEASE STATES AND CONDITIONS
Title (de)
ENANTIOMERENREINER GP-AGONIST ZUR VERWENDUNG BEI DER BEHANDLUNG VON KRANKHEITSZUSTÄNDEN UND ERKRANKUNGEN
Title (fr)
AGONISTE GPER PURIFIÉ DE MANIÈRE ÉNANTIOMÈRE DESTINÉ À L'UTILISATION DANS LE TRAITEMENT D'ÉTATS ET D'AFFECTATIONS PATHOLOGIQUES
Publication
Application
Priority
- US 2019042827 W 20190722
- US 201862701726 P 20180721
Abstract (en)
[origin: US2020024262A1] The present disclosure provides 1) an enantiomerically purified compound SRR G-1, or a derivative thereof, including specific crystal forms, salts and co-crystals that modulates G protein-coupled estrogen receptor activity, 2) pharmaceutical and cosmetic compositions comprising an enantiomerically purified SRR G-1, or a derivative thereof, and 3) methods of treating or preventing disease states and conditions and cosmetic conditions mediated through these receptors and related methods thereof in humans and animals.
IPC 8 full level
C07D 405/04 (2006.01); A61K 31/47 (2006.01); A61P 35/00 (2006.01); C07C 309/19 (2006.01); C07C 309/29 (2006.01); C07C 309/35 (2006.01)
CPC (source: EP IL KR US)
A61K 31/473 (2013.01 - KR); A61P 3/10 (2018.01 - KR); A61P 15/18 (2018.01 - KR); A61P 17/00 (2018.01 - KR); A61P 35/00 (2018.01 - EP KR); C07C 309/19 (2013.01 - EP); C07C 309/29 (2013.01 - EP); C07C 309/35 (2013.01 - EP); C07D 405/04 (2013.01 - EP IL KR US); C07B 2200/07 (2013.01 - EP IL KR US); C07B 2200/13 (2013.01 - EP IL KR US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
US 2020024262 A1 20200123; AU 2019310029 A1 20210204; BR 112021001031 A2 20210413; CA 3107109 A1 20200130; CN 112469409 A 20210309; DK 3823617 T3 20240603; EP 3823617 A1 20210526; EP 3823617 A4 20220420; EP 3823617 B1 20240306; EP 4356913 A2 20240424; FI 3823617 T3 20240529; IL 280283 A 20210301; IL 280283 B1 20240601; JP 2021532148 A 20211125; KR 20210049778 A 20210506; MX 2021000809 A 20210615; US 10934277 B2 20210302; US 11760749 B2 20230919; US 2020140417 A1 20200507; US 2022033385 A1 20220203; US 2022089576 A1 20220324; US 2023382896 A1 20231130; WO 2020023391 A1 20200130
DOCDB simple family (application)
US 201916518516 A 20190722; AU 2019310029 A 20190722; BR 112021001031 A 20190722; CA 3107109 A 20190722; CN 201980048925 A 20190722; DK 19842049 T 20190722; EP 19842049 A 20190722; EP 24161261 A 20190722; FI 19842049 T 20190722; IL 28028321 A 20210119; JP 2021504360 A 20190722; KR 20217002117 A 20190722; MX 2021000809 A 20190722; US 2019042827 W 20190722; US 201916682821 A 20191113; US 202117184870 A 20210225; US 202117328590 A 20210524; US 202318364690 A 20230803