EP 3870243 A1 20210901 - MARKING PRECURSOR WITH SQUARIC ACID COUPLING
Title (en)
MARKING PRECURSOR WITH SQUARIC ACID COUPLING
Title (de)
MARKIERUNGSVORLÄUFER MIT QUADRATSÄURE-KOPPLUNG
Title (fr)
PRÉCURSEUR DE MARQUAGE COMPRENANT UN COUPLAGE PAR ACIDE QUADRATIQUE
Publication
Application
Priority
- DE 102018126558 A 20181024
- EP 2019078614 W 20191021
Abstract (en)
[origin: WO2020083853A1] The invention relates to a marking precursor comprising a chelator or fluorination group for radiolabelling with 44Sc, 47Sc, 55Co, 62Cu, 64Cu, 67Cu, 66Ga, 67Ga, 68Ga, 89Zr, 86Y, 90Y, 90Nb, 99mTc, 111ln, 135Sm, 140Pr, 159Gd, 149Tb, 160Tb, 161Tb, 165Er, 166Dy, 166Ho, 175Yb, 177Lu, 186Re, 188Re, 213Bi and 225Ac or with 18F, 131I or 211At, and one or two biological targeting vectors which are coupled to the chelator or fluorinating group via one or more squaric acid groups. Formula (I).
IPC 8 full level
A61K 51/04 (2006.01); A61K 101/02 (2006.01); A61K 103/00 (2006.01); A61K 103/10 (2006.01); A61K 103/30 (2006.01); A61K 103/40 (2006.01)
CPC (source: CN EP KR US)
A61K 47/54 (2017.07 - US); A61K 51/0402 (2013.01 - EP); A61K 51/0446 (2013.01 - EP KR); A61K 51/0455 (2013.01 - EP KR); A61K 51/0478 (2013.01 - US); A61K 51/0482 (2013.01 - CN US); A61K 51/0489 (2013.01 - EP KR); A61K 51/0497 (2013.01 - EP KR US); C07C 275/16 (2013.01 - EP KR); C07C 323/60 (2013.01 - EP KR); C07D 245/02 (2013.01 - EP KR); C07D 253/02 (2013.01 - EP KR); C07D 257/02 (2013.01 - EP KR); C07D 401/14 (2013.01 - CN EP KR); C07D 403/12 (2013.01 - EP KR); C07F 5/025 (2013.01 - EP KR); C07F 9/3808 (2013.01 - EP KR); C07F 9/3873 (2013.01 - EP KR); C07F 9/6506 (2013.01 - EP KR); C07F 9/6515 (2013.01 - EP KR); C07F 9/65583 (2013.01 - EP KR); C07B 2200/05 (2013.01 - EP KR); C07C 2601/04 (2017.04 - EP KR)
Citation (search report)
See references of WO 2020083853A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2020083853 A1 20200430; AU 2019365377 A1 20210429; BR 112021007659 A2 20210727; CA 3116272 A1 20200430; CN 113164630 A 20210723; CN 114796533 A 20220729; CN 114796533 B 20240126; DE 102018126558 A1 20200430; EP 3870243 A1 20210901; EP 4082581 A1 20221102; JP 2022509385 A 20220120; KR 20210083289 A 20210706; US 11833229 B2 20231205; US 2021369877 A1 20211202; US 2022331456 A1 20221020
DOCDB simple family (application)
EP 2019078614 W 20191021; AU 2019365377 A 20191021; BR 112021007659 A 20191021; CA 3116272 A 20191021; CN 201980070046 A 20191021; CN 202210533888 A 20191021; DE 102018126558 A 20181024; EP 19800930 A 20191021; EP 22174349 A 20191021; JP 2021547891 A 20191021; KR 20217015486 A 20191021; US 201917287692 A 20191021; US 202217745100 A 20220516