EP 3906253 A1 20211110 - CONOTOXIN PEPTIDE ANALOGS AND USES FOR THE TREATMENT OF PAIN AND INFLAMMATORY CONDITIONS
Title (en)
CONOTOXIN PEPTIDE ANALOGS AND USES FOR THE TREATMENT OF PAIN AND INFLAMMATORY CONDITIONS
Title (de)
CONOTOXIN-PEPTIDANALOGA UND VERWENDUNGEN ZUR BEHANDLUNG VON SCHMERZEN UND ENTZÜNDLICHEN ZUSTÄNDEN
Title (fr)
ANALOGUES PEPTIDIQUES DE CONOTOXINE ET LEURS UTILISATIONS POUR LE TRAITEMENT DE LA DOULEUR ET D'AFFECTIONS INFLAMMATOIRES
Publication
Application
Priority
US 2019012307 W 20190104
Abstract (en)
[origin: WO2020142102A1] Provided herein are alpha-conotoxin peptide analogs, including alpha-conotoxin peptide analogs that are covalently attached to polyethylene glycol (PEG), and pharmaceutical compositions of such alpha-conotoxin peptide analogs. Also provided herein are methods of treating or preventing a condition conducive to treatment or prevention by inhibition of an a9- containing nicotinic acetylcholine receptor (nAChR) (e.g., the α9α10 subtype of the nAChR) in a subject.
IPC 8 full level
C07K 14/435 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP IL KR)
A61K 38/00 (2013.01 - IL); A61K 38/1767 (2013.01 - KR); A61K 47/60 (2017.07 - EP IL KR); C07K 7/08 (2013.01 - EP IL KR); C07K 14/43504 (2013.01 - EP IL KR); A61K 38/00 (2013.01 - EP)
Citation (search report)
See references of WO 2020142102A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2020142102 A1 20200709; WO 2020142102 A9 20201119; AU 2019418319 A1 20210722; BR 112021013302 A2 20210914; CA 3125383 A1 20200709; CL 2021001775 A1 20220527; CN 113966339 A 20220121; CO 2021008845 A2 20211029; CR 20210363 A 20211210; EP 3906253 A1 20211110; IL 284574 A 20210831; JP 2022522935 A 20220421; KR 20210116505 A 20210927; MX 2021008070 A 20211013; PE 20211734 A1 20210906; SG 11202106847S A 20210729
DOCDB simple family (application)
US 2019012307 W 20190104; AU 2019418319 A 20190104; BR 112021013302 A 20190104; CA 3125383 A 20190104; CL 2021001775 A 20210702; CN 201980093540 A 20190104; CO 2021008845 A 20210702; CR 20210363 A 20190104; EP 19702500 A 20190104; IL 28457421 A 20210702; JP 2021538994 A 20190104; KR 20217024613 A 20190104; MX 2021008070 A 20190104; PE 2021001115 A 20190104; SG 11202106847S A 20190104