EP 3969457 A4 20230524 - METHODS OF PREPARING MACROCYCLIC INDOLES
Title (en)
METHODS OF PREPARING MACROCYCLIC INDOLES
Title (de)
VERFAHREN ZUR HERSTELLUNG MAKROCYCLISCHER INDOLE
Title (fr)
PROCÉDÉS DE PRÉPARATION D'INDOLES MACROCYCLIQUES
Publication
Application
Priority
- US 201962849515 P 20190517
- US 2020033067 W 20200515
Abstract (en)
[origin: WO2020236556A1] The present invention relates to methods of preparing substituted indole derivatives of general formula (I) : in which R1, R2, R3, R4, R5, R6, A and L are as defined herein, and intermediate compounds useful for preparing said compounds. These compounds are useful for manufacturing pharmaceutical compositions for the treatment or prophylaxis of diseases, in particular of hyperproliferative disorders, as a sole agent or in combination with other active ingredients.
IPC 8 full level
C07D 498/14 (2006.01); C07D 413/00 (2006.01); C07D 413/14 (2006.01)
CPC (source: EP US)
C07D 403/04 (2013.01 - EP US); C07D 498/16 (2013.01 - EP US)
Citation (search report)
No further relevant documents disclosed
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
WO 2020236556 A1 20201126; CN 114127079 A 20220301; EP 3969457 A1 20220323; EP 3969457 A4 20230524; US 2022289762 A1 20220915
DOCDB simple family (application)
US 2020033067 W 20200515; CN 202080050407 A 20200515; EP 20808660 A 20200515; US 202017612019 A 20200515