Global Patent Index - EP 3986405 A4

EP 3986405 A4 20230614 - COMPOUNDS FOR INHIBITING FGFR4

Title (en)

COMPOUNDS FOR INHIBITING FGFR4

Title (de)

VERBINDUNGEN ZUR HEMMUNG VON FGFR4

Title (fr)

COMPOSÉS POUR INHIBER FGFR4

Publication

EP 3986405 A4 20230614 (EN)

Application

EP 20825842 A 20200618

Priority

  • US 201962864883 P 20190621
  • US 2020038541 W 20200618

Abstract (en)

[origin: WO2020257527A1] Provided herein are compounds which inhibit FGFR4, compositions thereof, methods of their preparation, and methods for treating disorders mediated by FGFR4 such as cancer.

IPC 8 full level

C07D 471/04 (2006.01); A61K 31/4375 (2006.01); A61K 31/517 (2006.01); A61K 31/519 (2006.01); A61P 35/00 (2006.01)

CPC (source: EP US)

A61K 31/44 (2013.01 - EP US); A61K 31/4545 (2013.01 - EP); A61K 31/47 (2013.01 - EP US); A61K 31/506 (2013.01 - EP US); A61K 39/3955 (2013.01 - US); C07D 471/04 (2013.01 - EP US); A61P 35/00 (2018.01 - EP)

C-Set (source: EP)

  1. A61K 31/4545 + A61K 2300/00
  2. A61K 31/506 + A61K 2300/00
  3. A61K 31/47 + A61K 2300/00
  4. A61K 31/44 + A61K 2300/00

Citation (search report)

  • [A] WO 2015059668 A1 20150430 - NOVARTIS AG [CH], et al
  • [A] WO 2017164705 A1 20170928 - DAEGU-GYEONGBUK MEDICAL INNOVATION FOUND [KR], et al
  • [Y] EP 3444250 A1 20190220 - JIANGSU HANSOH PHARMACEUTICAL GROUP CO LTD [CN], et al
  • [Y] THOMAS KNOEPFEL ET AL: "2-Formylpyridyl Ureas as Highly Selective Reversible-Covalent Inhibitors of Fibroblast Growth Factor Receptor 4", ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, no. 3, 1 February 2018 (2018-02-01), US, pages 215 - 220, XP055584418, ISSN: 1948-5875, DOI: 10.1021/acsmedchemlett.7b00485
  • See also references of WO 2020257527A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2020257527 A1 20201224; AU 2020298246 A1 20220127; CA 3144366 A1 20201224; CN 114144176 A 20220304; EP 3986405 A1 20220427; EP 3986405 A4 20230614; JP 2022537415 A 20220825; US 2022362245 A1 20221117

DOCDB simple family (application)

US 2020038541 W 20200618; AU 2020298246 A 20200618; CA 3144366 A 20200618; CN 202080052789 A 20200618; EP 20825842 A 20200618; JP 2021576063 A 20200618; US 202017621203 A 20200618