EP 3986405 A4 20230614 - COMPOUNDS FOR INHIBITING FGFR4
Title (en)
COMPOUNDS FOR INHIBITING FGFR4
Title (de)
VERBINDUNGEN ZUR HEMMUNG VON FGFR4
Title (fr)
COMPOSÉS POUR INHIBER FGFR4
Publication
Application
Priority
- US 201962864883 P 20190621
- US 2020038541 W 20200618
Abstract (en)
[origin: WO2020257527A1] Provided herein are compounds which inhibit FGFR4, compositions thereof, methods of their preparation, and methods for treating disorders mediated by FGFR4 such as cancer.
IPC 8 full level
C07D 471/04 (2006.01); A61K 31/4375 (2006.01); A61K 31/517 (2006.01); A61K 31/519 (2006.01); A61P 35/00 (2006.01)
CPC (source: EP US)
A61K 31/44 (2013.01 - EP US); A61K 31/4545 (2013.01 - EP); A61K 31/47 (2013.01 - EP US); A61K 31/506 (2013.01 - EP US); A61K 39/3955 (2013.01 - US); C07D 471/04 (2013.01 - EP US); A61P 35/00 (2018.01 - EP)
C-Set (source: EP)
Citation (search report)
- [A] WO 2015059668 A1 20150430 - NOVARTIS AG [CH], et al
- [A] WO 2017164705 A1 20170928 - DAEGU-GYEONGBUK MEDICAL INNOVATION FOUND [KR], et al
- [Y] EP 3444250 A1 20190220 - JIANGSU HANSOH PHARMACEUTICAL GROUP CO LTD [CN], et al
- [Y] THOMAS KNOEPFEL ET AL: "2-Formylpyridyl Ureas as Highly Selective Reversible-Covalent Inhibitors of Fibroblast Growth Factor Receptor 4", ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, no. 3, 1 February 2018 (2018-02-01), US, pages 215 - 220, XP055584418, ISSN: 1948-5875, DOI: 10.1021/acsmedchemlett.7b00485
- See also references of WO 2020257527A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
WO 2020257527 A1 20201224; AU 2020298246 A1 20220127; CA 3144366 A1 20201224; CN 114144176 A 20220304; EP 3986405 A1 20220427; EP 3986405 A4 20230614; JP 2022537415 A 20220825; US 2022362245 A1 20221117
DOCDB simple family (application)
US 2020038541 W 20200618; AU 2020298246 A 20200618; CA 3144366 A 20200618; CN 202080052789 A 20200618; EP 20825842 A 20200618; JP 2021576063 A 20200618; US 202017621203 A 20200618