EP 4076659 A1 20221026 - MACROCYCLIC AMIDES ACTING AS PLASMEPSIN INHBITORS FOR THE TREATMENT OF MALARIA
Title (en)
MACROCYCLIC AMIDES ACTING AS PLASMEPSIN INHBITORS FOR THE TREATMENT OF MALARIA
Title (de)
MAKROZYKLISCHE AMIDE ALS PLASMEPSIN-INHIBITOREN FÜR DIE BEHANDLUNG VON MALARIA
Title (fr)
AMIDES MACROCYCLIQUES AGISSANT COMME INHIBITEURS DE LA PLASMEPSINE POUR LE TRAITEMENT DU PALUDISME
Publication
Application
Priority
IB 2019061066 W 20191219
Abstract (en)
[origin: WO2021123883A1] The present invention relates to medicine and in particular to the treatment of malarial infections, more particularly to inhibitors of malarial aspartic proteases - plasmepsins. Even more particularly, the invention relates to macrocyclic amides and pharmaceutical compositions thereof and their use as inhibitors for plasmepsins (Plm).
IPC 8 full level
A61P 33/06 (2006.01); A61K 31/33 (2006.01); C07D 498/08 (2006.01)
CPC (source: EP)
A61P 33/06 (2017.12); C07D 498/08 (2013.01); Y02A 50/30 (2017.12)
Citation (search report)
See references of WO 2021123883A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
Designated validation state (EPC)
KH MA MD TN
DOCDB simple family (publication)
DOCDB simple family (application)
IB 2019061066 W 20191219; EP 19835811 A 20191219