Global Patent Index - EP 4095136 A1

EP 4095136 A1 20221130 - SYNTHESIS AND USE OF CLASS OF RESPIRATORY SYNCYTIAL VIRUS INHIBITORS

Title (en)

SYNTHESIS AND USE OF CLASS OF RESPIRATORY SYNCYTIAL VIRUS INHIBITORS

Title (de)

SYNTHESE UND VERWENDUNG EINER KLASSE VON RESPIRATORISCHEN SYNCYTIALVIRUS-INHIBITOREN

Title (fr)

SYNTHÈSE ET UTILISATION D'UNE CLASSE D'INHIBITEURS DU VIRUS RESPIRATOIRE SYNCYTIAL

Publication

EP 4095136 A1 20221130 (EN)

Application

EP 21744323 A 20210121

Priority

  • CN 202010075139 A 20200122
  • CN 2021073042 W 20210121

Abstract (en)

The present disclosure provides the synthesis and application of respiratory syncytial virus inhibitor, being a compound of formula I or a pharmaceutically acceptable salt, ester, isomer, solvate, prodrug or isotope label thereof.Compared with the existing inhibitors, the compounds of formula I have the advantages of superior activity and higher exposure in vivo.

IPC 8 full level

C07D 417/14 (2006.01); A61K 31/554 (2006.01); A61P 11/00 (2006.01); A61P 31/14 (2006.01); C07D 417/04 (2006.01)

CPC (source: CN EP KR US)

A61K 31/554 (2013.01 - CN KR US); A61P 11/00 (2017.12 - EP KR); A61P 31/12 (2017.12 - CN EP); A61P 31/14 (2017.12 - EP KR US); C07D 417/04 (2013.01 - CN EP KR); C07D 417/14 (2013.01 - EP KR); C07D 487/10 (2013.01 - KR)

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

Designated validation state (EPC)

KH MA MD TN

DOCDB simple family (publication)

EP 4095136 A1 20221130; EP 4095136 A4 20230705; CN 113149977 A 20210723; CN 115023423 A 20220906; JP 2023511152 A 20230316; KR 20220130761 A 20220927; US 2023090060 A1 20230323; WO 2021147947 A1 20210729

DOCDB simple family (application)

EP 21744323 A 20210121; CN 202010075139 A 20200122; CN 2021073042 W 20210121; CN 202180010637 A 20210121; JP 2022544247 A 20210121; KR 20227028783 A 20210121; US 202117790987 A 20210121