Global Patent Index - EP 4100125 A1

EP 4100125 A1 20221214 - POLYMORPH OF RUCAPARIB MESYLATE

Title (en)

POLYMORPH OF RUCAPARIB MESYLATE

Title (de)

POLYMORPH VON RUCAPARIB-MESYLAT

Title (fr)

POLYMORPHE DE MÉSYLATE DE RUCAPARIB

Publication

EP 4100125 A1 20221214 (EN)

Application

EP 21702480 A 20210128

Priority

  • EP 20155091 A 20200203
  • EP 2021052029 W 20210128

Abstract (en)

[origin: WO2021156140A1] The present invention relates to an anhydrous crystalline form of rucaparib mesylate, preferably in polymorphically pure form and to a process for its preparation. Furthermore, the invention relates to a pharmaceutical composition comprising the anhydrous crystalline form of rucaparib mesylate, preferably in polymorphically pure form and at least one pharmaceutically acceptable excipient. The pharmaceutical composition of the present invention can be used as a medicament, in particular for the treatment of cancer.

IPC 8 full level

A61P 35/00 (2006.01); A61K 31/55 (2006.01); C07D 487/06 (2006.01)

CPC (source: EP)

A61P 35/00 (2017.12); C07D 487/06 (2013.01)

Citation (search report)

See references of WO 2021156140A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

Designated validation state (EPC)

KH MA MD TN

DOCDB simple family (publication)

WO 2021156140 A1 20210812; EP 4100125 A1 20221214

DOCDB simple family (application)

EP 2021052029 W 20210128; EP 21702480 A 20210128