EP 4229033 A1 20230823 - PROCESSES OF PREPARING 3-FLUORO-5-(((1S,2AR)-1,3,3,4,4-PENTAFLUORO-2A-HYDROXY-2,2A,3,4-TETRAHYDRO-1H-CYCLOPENTA[CD]INDEN-7-YL)OXY)-BENZONITRILE
Title (en)
PROCESSES OF PREPARING 3-FLUORO-5-(((1S,2AR)-1,3,3,4,4-PENTAFLUORO-2A-HYDROXY-2,2A,3,4-TETRAHYDRO-1H-CYCLOPENTA[CD]INDEN-7-YL)OXY)-BENZONITRILE
Title (de)
VERFAHREN ZUR HERSTELLUNG VON 3-FLUOR-5-((1S,2AR)-1,3,3,4,4-PENTAFLUOR-2A-HYDROXY-2,2A,3,4-TETRAHYDRO-1H-CYCLOPENTA[CD!INDEN-7-YL)OXY)-BENZONITRIL
Title (fr)
PROCÉDÉS DE PRÉPARATION DE 3-FLUORO-5-(((1S,2AR)-1,3,3,4,4-PENTAFLUORO-2A-HYDROXY-2,2A,3,4-TÉTRAHYDRO-1H-CYCLOPENTA[CD]INDEN-7-YL)OXY)-BENZONITRILE
Publication
Application
Priority
- CN 2020121745 W 20201019
- US 2021055295 W 20211015
Abstract (en)
[origin: WO2022086822A1] Disclosed herein are processes for preparing 3-fluoro-5-(((1S,2aR)-1,3,3,4,4-pentafluoro-2a-hydroxy-2,2a,3,4-tetrahydro-1H-cyclopenta[cd]inden-7-yl)oxy)benzonitrile or a pharmaceutically acceptable salt thereof.
IPC 8 full level
C07C 253/30 (2006.01); C07C 29/38 (2006.01); C07C 29/62 (2006.01); C07C 35/32 (2006.01); C07C 35/52 (2006.01); C07C 255/54 (2006.01)
CPC (source: EP IL KR)
C07C 29/38 (2013.01 - EP IL KR); C07C 29/58 (2013.01 - KR); C07C 29/62 (2013.01 - EP IL KR); C07C 35/32 (2013.01 - IL KR); C07C 35/52 (2013.01 - IL KR); C07C 45/40 (2013.01 - EP IL KR); C07C 45/673 (2013.01 - EP IL KR); C07C 49/737 (2013.01 - IL KR); C07C 253/30 (2013.01 - EP IL KR); C07C 255/54 (2013.01 - IL KR); C07B 2200/07 (2013.01 - EP IL KR); C07C 2602/08 (2017.05 - EP IL KR); C07C 2603/10 (2017.05 - EP IL KR)
C-Set (source: EP)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
Designated validation state (EPC)
KH MA MD TN
DOCDB simple family (publication)
WO 2022086822 A1 20220428; AU 2021364337 A1 20230601; CA 3197932 A1 20220428; CN 116507601 A 20230728; EP 4229033 A1 20230823; IL 301897 A 20230601; JP 2023548666 A 20231120; KR 20230092936 A 20230626; TW 202233569 A 20220901; WO 2022082329 A1 20220428
DOCDB simple family (application)
US 2021055295 W 20211015; AU 2021364337 A 20211015; CA 3197932 A 20211015; CN 2020121745 W 20201019; CN 202180070640 A 20211015; EP 21805779 A 20211015; IL 30189723 A 20230403; JP 2023522392 A 20211015; KR 20237015120 A 20211015; TW 110138778 A 20211019