EP 4294798 A1 20231227 - FACTOR XIIA INHIBITORS
Title (en)
FACTOR XIIA INHIBITORS
Title (de)
FAKTOR XIIA-HEMMER
Title (fr)
INHIBITEURS DU FACTEUR XIIA
Publication
Application
Priority
- GB 202102384 A 20210219
- US 202163151178 P 20210219
- GB 202104788 A 20210401
- US 202163169607 P 20210401
- GB 202106284 A 20210430
- US 202163182283 P 20210430
- GB 2022050447 W 20220218
Abstract (en)
[origin: WO2022175675A1] The present invention provides compounds of formula (I): compositions comprising such compounds; the use of such compounds in medicine; and methods of treating patients with such compounds; wherein A, W, V, Z, U, X, Y and B are as defined herein.
IPC 8 full level
C07D 401/12 (2006.01); A61K 31/437 (2006.01); A61K 31/4725 (2006.01); A61K 31/4985 (2006.01); A61K 31/4995 (2006.01); A61K 31/506 (2006.01); A61P 7/02 (2006.01); A61P 7/10 (2006.01); A61P 9/00 (2006.01); C07D 401/14 (2006.01); C07D 405/12 (2006.01); C07D 413/14 (2006.01); C07D 471/04 (2006.01); C07D 487/04 (2006.01); C07D 487/08 (2006.01); C07D 519/00 (2006.01)
CPC (source: EP IL KR)
A61K 31/4725 (2013.01 - KR); A61P 7/02 (2018.01 - EP IL KR); A61P 7/10 (2018.01 - EP IL KR); A61P 9/00 (2018.01 - EP IL); C07D 401/12 (2013.01 - EP IL KR); C07D 401/14 (2013.01 - EP IL KR); C07D 405/12 (2013.01 - EP IL KR); C07D 405/14 (2013.01 - KR); C07D 413/14 (2013.01 - EP IL KR); C07D 471/04 (2013.01 - EP IL KR); C07D 487/04 (2013.01 - EP IL KR); C07D 487/08 (2013.01 - EP IL KR); C07D 519/00 (2013.01 - EP IL)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
Designated validation state (EPC)
KH MA MD TN
DOCDB simple family (publication)
WO 2022175675 A1 20220825; AU 2022222458 A1 20230824; BR 112023016539 A2 20231114; CA 3211159 A1 20220825; CL 2023002446 A1 20240112; CO 2023012342 A2 20230929; EP 4294798 A1 20231227; IL 305307 A 20231001; JP 2024507222 A 20240216; KR 20230157981 A 20231117; MX 2023009677 A 20230825; TW 202302565 A 20230116
DOCDB simple family (application)
GB 2022050447 W 20220218; AU 2022222458 A 20220218; BR 112023016539 A 20220218; CA 3211159 A 20220218; CL 2023002446 A 20230817; CO 2023012342 A 20230918; EP 22706887 A 20220218; IL 30530723 A 20230817; JP 2023550048 A 20220218; KR 20237032029 A 20220218; MX 2023009677 A 20220218; TW 111106094 A 20220218