Global Patent Index - EP 4313992 A1

EP 4313992 A1 20240207 - POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE

Title (en)

POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE

Title (de)

POLYMORPHE FORMEN VON (S)-12-FLUOR-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4)TRIAZOLO[4',3':1,6,7PYRIDO[3,2-B!BENZOFURO[4,3-FG [1,4)OXNIN

Title (fr)

FORMES POLYMORPHES DE (S)-12-FLUORO-4-(1-MÉTHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TÉTRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE

Publication

EP 4313992 A1 20240207 (EN)

Application

EP 22718451 A 20220331

Priority

  • US 202163170226 P 20210402
  • US 2022022895 W 20220331

Abstract (en)

[origin: WO2022212748A1] The disclosure is in part directed to crystalline forms of (S)-12-fluoro-4-(1-methyl-1H-pyrazol-5-yl)-7a,8,13,14-tetrahydro-7H-[1,2,4]triazolo[4',3':1,6]pyrido[3,2-b]benzofuro[4,3-fg][1,4]oxazonine.

IPC 8 full level

C07D 491/22 (2006.01); A61K 31/5365 (2006.01); A61P 35/00 (2006.01)

CPC (source: EP US)

A61K 31/437 (2013.01 - US); A61P 35/00 (2018.01 - EP); C07D 491/22 (2013.01 - EP); C07D 498/22 (2013.01 - US)

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

Designated validation state (EPC)

KH MA MD TN

DOCDB simple family (publication)

WO 2022212748 A1 20221006; EP 4313992 A1 20240207; US 2024199645 A1 20240620

DOCDB simple family (application)

US 2022022895 W 20220331; EP 22718451 A 20220331; US 202218553352 A 20220331