EP 4313992 A1 20240207 - POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE
Title (en)
POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE
Title (de)
POLYMORPHE FORMEN VON (S)-12-FLUOR-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4)TRIAZOLO[4',3':1,6,7PYRIDO[3,2-B!BENZOFURO[4,3-FG [1,4)OXNIN
Title (fr)
FORMES POLYMORPHES DE (S)-12-FLUORO-4-(1-MÉTHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TÉTRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE
Publication
Application
Priority
- US 202163170226 P 20210402
- US 2022022895 W 20220331
Abstract (en)
[origin: WO2022212748A1] The disclosure is in part directed to crystalline forms of (S)-12-fluoro-4-(1-methyl-1H-pyrazol-5-yl)-7a,8,13,14-tetrahydro-7H-[1,2,4]triazolo[4',3':1,6]pyrido[3,2-b]benzofuro[4,3-fg][1,4]oxazonine.
IPC 8 full level
C07D 491/22 (2006.01); A61K 31/5365 (2006.01); A61P 35/00 (2006.01)
CPC (source: EP US)
A61K 31/437 (2013.01 - US); A61P 35/00 (2018.01 - EP); C07D 491/22 (2013.01 - EP); C07D 498/22 (2013.01 - US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
Designated validation state (EPC)
KH MA MD TN
DOCDB simple family (publication)
WO 2022212748 A1 20221006; EP 4313992 A1 20240207; US 2024199645 A1 20240620
DOCDB simple family (application)
US 2022022895 W 20220331; EP 22718451 A 20220331; US 202218553352 A 20220331