Global Patent Index - EP 4400495 A1

EP 4400495 A1 20240717 - DOPAMINE D3/D2 RECEPTOR MODULATING COMPOUNDS

Title (en)

DOPAMINE D3/D2 RECEPTOR MODULATING COMPOUNDS

Title (de)

DOPAMIN-D3/D2-REZEPTOR-MODULIERENDE VERBINDUNGEN

Title (fr)

COMPOSÉS MODULANT LE RÉCEPTEUR D3/D2 DE LA DOPAMINE

Publication

EP 4400495 A1 20240717 (EN)

Application

EP 24151077 A 20240110

Priority

US 202363479530 P 20230111

Abstract (en)

The present disclosure provides for compounds of Formula (I):wherein R<sup>1</sup> has any of the values defined in the specification, and pharmaceutically acceptable salts thereof, that are useful as agents in the treatment of diseases and conditions including schizophrenia. Also provided are pharmaceutical compositions comprising compounds of Formula (I).

IPC 8 full level

C07D 295/155 (2006.01); A61P 25/18 (2006.01)

CPC (source: EP KR)

A61K 31/495 (2013.01 - KR); A61P 25/18 (2018.01 - EP KR); C07D 295/135 (2013.01 - KR); C07D 295/155 (2013.01 - EP)

Citation (applicant)

  • WO 2010070370 A1 20100624 - RICHTER GEDEON NYRT [HU], et al
  • WO 2005012266 A1 20050210 - RICHTER GEDEON VEGYESZET [HU], et al
  • SOKOLOFF, P. ET AL., NATURE, vol. 347, 1990, pages 146
  • SCHWARTZ, J.-C. ET AL., CLIN. NEUROPHARMACOLOGY., vol. 16, 1993, pages 295
  • "GenBank", Database accession no. U32499

Citation (search report)

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC ME MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA

Designated validation state (EPC)

KH MA MD TN

DOCDB simple family (publication)

EP 4400495 A1 20240717; JP 2024098972 A 20240724; KR 20240112213 A 20240718; WO 2024150068 A2 20240718; WO 2024150068 A3 20240822

DOCDB simple family (application)

EP 24151077 A 20240110; IB 2024000026 W 20240110; JP 2024001696 A 20240110; KR 20240002897 A 20240108