(19)
(11)EP 3 807 251 A1

(12)

(43)Date of publication:
21.04.2021 Bulletin 2021/16

(21)Application number: 19758804.9

(22)Date of filing:  17.06.2019
(51)International Patent Classification (IPC): 
C07D 233/66(2006.01)
A61P 29/00(2006.01)
C07D 401/04(2006.01)
A61K 31/4178(2006.01)
(86)International application number:
PCT/IB2019/055045
(87)International publication number:
WO 2019/244000 (26.12.2019 Gazette  2019/52)
(84)Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30)Priority: 18.06.2018 US 201862686323 P

(71)Applicant: Janssen Pharmaceutica NV
2340 Beerse (BE)

(72)Inventors:
  • MARTIN, Connor L.
    San Diego, California 92121 (US)
  • FENNEMA, Elizabeth G.
    San Diego, California 92121 (US)
  • KUMMER, David A.
    San Diego, California 92121 (US)
  • NISHIMURA, Rachel T.
    San Diego, California 92121 (US)
  • TANIS, Virginia M.
    San Diego, California 92121 (US)
  • WOODS, Craig R.
    San Diego, California 92121 (US)
  • FOURIE, Anne M.
    San Diego, California 92121 (US)
  • XUE, Xiaohua
    San Diego, California 92121 (US)
  • GOLDBERG, Steven
    San Diego, California 92121 (US)

(74)Representative: Warner, James Alexander 
Carpmaels & Ransford LLP One Southampton Row
London WC1B 5HA
London WC1B 5HA (GB)

  


(54)PHENYL AND PYRIDINYL SUBSTITUTED IMIDAZOLES AS MODULATORS OF RORYT