(19)
(11)EP 2 705 033 A1

(12)

(43)Date of publication:
12.03.2014 Bulletin 2014/11

(21)Application number: 12717736.8

(22)Date of filing:  30.04.2012
(51)International Patent Classification (IPC): 
C07D 403/12(2006.01)
A61K 31/497(2006.01)
A61K 31/4155(2006.01)
A61P 3/10(2006.01)
(86)International application number:
PCT/EP2012/057876
(87)International publication number:
WO 2012/150202 (08.11.2012 Gazette  2012/45)
(84)Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

(30)Priority: 03.05.2011 US 201161481789 P

(71)Applicant: F. Hoffmann-La Roche AG
4070 Basel (CH)

(72)Inventors:
  • BERTHEL, Steven Joseph
    Mendham Township, NJ 07945 (US)
  • KESTER, Robert Francis
    West Orange, NJ 07052 (US)
  • ORZECHOWSKI, Lucja
    Kinnelon, NJ 07405 (US)

(74)Representative: Salud, Carlos E. et al
F. Hoffmann-La Roche AG Patent Department Grenzacherstrasse 124
4070 Basel
4070 Basel (CH)

  


(54)ISOINDOLINONE DERIVATIVES