(19)
(11)EP 1 399 146 A1

(12)

(43)Date of publication:
24.03.2004 Bulletin 2004/13

(21)Application number: 02739721.5

(22)Date of filing:  04.06.2002
(51)International Patent Classification (IPC)7A61K 31/277, C07C 255/42
(86)International application number:
PCT/US2002/017922
(87)International publication number:
WO 2002/098406 (12.12.2002 Gazette  2002/50)
(84)Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30)Priority: 04.06.2001 US 295744 P

(71)Applicant: AXYS PHARMACEUTICALS, INC.
South San Francisco, CA 94080 (US)

(72)Inventors:
  • PATTERSON, John, W.
    Mountain View, CA 94040 (US)
  • ZIPFEL, Sheila
    Mountain Vlew, CA 9403 (US)

(74)Representative: Thomson, Paul Anthony 
Potts, Kerr & Co.,15, Hamilton Square
Birkenhead,Merseyside CH41 6BR
Birkenhead,Merseyside CH41 6BR (GB)

  


(54)NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS