(19)
(11)EP 1 278 759 A1

(12)

(43)Date of publication:
29.01.2003 Bulletin 2003/05

(21)Application number: 01935025.5

(22)Date of filing:  02.05.2001
(51)International Patent Classification (IPC)7C07F 9/24, A61K 31/664, A61P 35/04
(86)International application number:
PCT/US0114/290
(87)International publication number:
WO 0108/3496 (08.11.2001 Gazette  2001/45)
(84)Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30)Priority: 02.05.2000 US 563181

(71)Applicant: TELIK, INC.
South San Francisco, CA 94080 (US)

(72)Inventors:
  • HERR, Jason, R.
    Voorheesville, NY 12186 (US)
  • LUM, Robert, T.
    Palo Alto, CA 94306 (US)
  • SCHOW, Steven, R.
    Redwood Shores, CA 94065 (US)
  • MENG, Fanying
    San Francisco, CA 94122 (US)
  • KOZLOWSKI, Michael, R.
    Palo Alto, CA 94303 (US)
  • ZHICHKIN, Pavel
    Albany, NY 12208 (US)

(74)Representative: Barz, Peter, Dr. 
PatentanwaltKaiserplatz 2
80803 München
80803 München (DE)

  


(54)BIS-(N,N'-BIS-(2-HALOETHYL)AMINO) PHOSPHORAMIDATES AS ANTITUMOR AGENTS