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Irreversible Inhibition of Human Immunodeficiency Virus Type 1 Integrase by Dicaffeoylquinic Acids   [0179] 
Effects of nucleotide analogues on human immunodeficiency virus type 1 integrase   [0180] 
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Antiviral Research   [0207] 
Novel membrane-interactive ether lipid analogs that inhibit infectious HIV-1 production and induce defective virus formation   [0208] 
Synthesis and evaluation of novel ether lipid nucleoside conjugates for anti-HIV activity   [0208] 
Greatly enhanced inhibition of human immunodeficiency virus type 1 replication in CEM and HT4-6C cells by 3'-deoxythymidine diphosphate dimyristoylglycerol, a lipid prodrug of 3'-deoxythymidine   [0208] 
Synthesis and antiretroviral activity of phospholipid analogs of azidothymidine and other antiviral nucleosides   [0208] 
Distribution of Kinase and deaminase of 1β-D-arabinofuranosylcytosine in tissues of man and muse   [0210] 
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Synthesis and antitumor activity of 1β-D-arabino-furanosylcytosine conjugates of cortisol and cortisone   [0210] 
Nucleoside conjugates as potential antitumor agents. 3. Synthesis and antitumor activity of 1-(β-D-arabinofuranosyl)cytosine conjugates of corticosteroids and selected lipophilic alcohols   [0210] 
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Phosphatidylazidothymidine: mechanism of antiretroviral action in CEM cells   [0210] 
Antiviral activity of phosphatidyl-dideoxycytidine in hepatitis B-infected cells and enhanced hepatic uptake in mice   [0210] 
Phosphatidylazidothymidine and phosphatidyl-ddC: Assessment of uptake in mouse lymphoid tissues and antiviral activities in human immunodeficiency virus-infected cells and in rauscher leukemia virus-infected mice   [0210] 
Synthesis and biological properties of some cyclic phosphotriesters derived from 2'-deoxy-5-fluorouridine   [0210] 
Monophosphoric acid esters of 7-β-hydroxycholesterol and of pyrimidine nucleoside as potential antitumor agents: synthesis and preliminary evaluation of antitumor activity   [0210] 
Synthesis, properties, and biological activity of some nucleoside cyclic phosphoramidates   [0210] 
Synthesis of diribonucleoside phosph (P.fwdarw.N) amino acid derivatives   [0210] 
Alkylated cAMP derivatives; selective synthesis and biological activities   [0210] 
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Comparison of antiviral effects of zidovudine phosphoramidate and phosphorodiamidate derivatives against HIV and ULV in vitro   [0210] 
Antitumor activity and pharmacology of 1-β-D-arabinofuranosylcytosine -5'-stearylphosphate; an orally active derivative of 1-β-Darabinofuranosylcytosine   [0210] 
The effects of adenosine- and guanosine 3',5' phosphoric and acid benzyl esters on guinea-pig ventricular myocardium   [0210] 
Synthesis and biological evaluation of some cyclic phosphoramidate nucleoside derivatives   [0210] 
Synthesis of lipophilic phosphate triester derivatives of 5-fluorouridine an arabinocytidine as anticancer prodrugs   [0210] 
The metabolism of exogenously supplied nucleotides by Escherichia coli.   [0210] 
Synthesis and toxicological properties of three naturally occurring cyanoepithioalkanes   [0210] 
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Synthesis and biological evaluation of some phosphate triester derivatives of the anti-viral drug Ara   [0210] 
Synthesis and evaluation of some novel phosphoramidate derivatives of 3'-azido-3'-deoxythymidine (AZT) as anti-HIV compounds   [0210] 
Synthesis and anti-HIV activity of some novel substituted dialkyl phosphate derivatives of AZT and ddCyd   [0210] 
Synthesis of some novel dialkyl phosphate derivative of 3'-modified nucleosides as potential anti-AIDS drugs   [0210] 
Synthesis and anti-HIV activity of some haloalkyl phosphoramidate derivatives of 3'-azido-3'-deoxythylmidine (AZT); potent activity of the trichloroethyl methoxyalaninyl compound   [0210] 
Intracellular delivery of bioactive AZT nucleotides by aryl phosphate derivatives of AZT   [0210] 
Alkyl hydrogen phosphate derivatives of the anti-HIV agent AZT may be less toxic than the parent nucleoside analogue   [0211] 
Synthesis of purine nucleoside 3',5'-cyclic phosphoramidates   [0211] 
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Improved brain delivery of AZT using a glycosyl phosphotriester prodrug   [0211] 
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The question of chair-twist equilibria for the phosphate rings of nucleoside cyclic 3',5'-monophosphates. HNMR and x-ray crystallographic study of the diastereomers of thymidine phenyl cyclic 3',5'-monophosphate   [0211] 
New photoactivatable cyclic nucleotides produce intracellular jumps in cyclic AMP and cyclic GMP concentrations   [0211] 
Synthesis and transmembrane transport studies by NMR of a glucosyl phospholipid of thymidine   [0211] 
Treatment of myelodysplastic syndromes with orally administered 1-β-D-arabinouranosylcytosine -5' stearylphosphate   [0211] 
A dihydropyridine carrier system for sustained delivery of 2',3' dideoxynucleosides to the brain   [0211] 
Activity of BRL47923 and its oral prodrug, SB203657A against a rauscher murine leukemia virus infection in mice   [0211] 
Synthesis and evaluation of novel ether lipid nucleoside conjugates for anti-HIV-1 activity   [0211] 
Decomposition pathways of the mono- and bis(pivaloyloxymethyl) esters of azidothymidine-5'-monophosphate in cell extract and in tissue culture medium; an application of the 'on-line ISRP-cleaning HPLC technique   [0211] 
Cyclic AMP and cyclic GMP   [0211] 
Synthesis and antiherpes virus activity of phosphate an phosphonate derivatives of 9-[(1,3-dihydroxy-2-propoxy)methyl]guanine   [0211] 
Intracellular delivery of nucleoside monophosphate through a reductase-mediated activation process   [0211] 
Toxicological assessment and health standard ratings for ethylene sulfide in the industrial atmosphere   [0211] 
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The potential of nucleotide analogs as inhibitors of Retro viruses and tumors   [0211] 
Lipophilic 5'-(alkylphosphate) esters of 1-β-D-arabinofiiranosylcytosine and its N4-acyl and 2.2'-anhydro-3'-O-acyl derivatives as potential prodrugs   [0211] 
Increased sensitivity of the walker turnout towards aromatic nitrogen mustards carrying basic side chains following glucose pretreatment   [0211] 
Phospholipid-nucleoside conjugates. 3. Synthesis and preliminary biological evaluation of 1-β-D-arabinofuranosylcytosine 5'diphosphate [-], 2-diacylglycerols   [0211] 
The degradation of 5-iododeoxyuridine and 5-bromoethoxyuridine by serum from different sources and its consequences for the use of these compounds for incorporation into DNA   [0211] 
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Membrane-permeable dideoxyuridine 5'-monophosphate analogue inhibits human immunodeficiency virus infection   [0211] 
Oral bioavailability of PMEA from PMEA prodrugs in male Sprague-Dawley rats   [0211] 
A facile one-step synthesis of 5' phosphatidiylnucleosides by an enzymatic two-phase reaction   [0211] 
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Differential effects of antiretroviral nucleoside analogs on mitochondrial function in HepG2 cells   [0293] 
Antiviral activities and cellular toxicities of modified 2',3'-dideoxy-2',3'-didehydrocytidine analogs   [0293] 
Quantitation of dihydropyrimidine dehydrogenase expression by real-time reverse transcription polymerase chain reaction   [0293] 
Effect of enantiomeric and racemic nucleoside analogs on mitochondrial functions in HepG2 cells   [0293] 
Fialuridine and its metabolites inhibit DNA polymerase gamma at sites of multiple adjacent analog incorporation, decrease mtDNA abundance, and cause mitochondrial structural defects in cultured hepatoblasts   [0293] 
Differential effects of antiretroviral nucleoside analogs on mitochondrial function in HepG2 cells   [0293] 
Mechanism of anti-human immunodeficiency virus activity of beta-D-6-cyclopropylamino-2',3'-didehydro-2',3'-dideoxyguanosine   [0294] 
Toxicity of 3'-azido-3'-deoxythymidine and 9-(1,3-dihydroxy-2-propoxymethyl) guanine for normal human hepatopoietic progenitor cells in vitro   [0295] 
Comparison of Cytotoxicity of the (-) and (+) enantiomer of 2',3'-dideoxy-3'-thiacytidine in normal human bone marrow progenitor cells   [0295] 
Antimicrob. Agents Chemother.   [0296] 
Ribonucleoside analogue that blocks replication or bovine viral diarrhea and hepatitis C viruses in culture   [0299] 
A simple method or estimating fifty percent endpoints   [0299] 
Enantiomeric synthesis of D- and L-cyclopentenyl nucleosides and their antiviral activity against HIV and West Nile virus   [0300] 
Activity of T-1106 in a Hamster Model of Yellow Fever Virus Infection   [0301] 
A scintillation proximity assay for dengue virus NS5 2'-O-methyltransferase-kinetic and inhibition analyses   [0302] 
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Mechanism of action of a pestivirus antiviral compound   [0307] 
Mechanism of action of a pestivirus antiviral compound   [0311] 
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