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Determination of the biological activity and structure activity relationships of drugs based on the highly cytotoxic duocarmycins and CC-1065   [0296] 
Antibody-directed enzyme prodrug therapy: a promising approach for a selective treatment of cancer based on prodrugs and monoclonal antibodies   [0296] 
Synthesis and biological evaluation of a novel pentagastrin-toxin conjugate designed for a targeted prodrug mono-therapy of cancer   [0296] 
Novel analogues of CC-1065 and the duocarmycins for the use in targeted tumour therapies   [0296] 
Synthesis and biological studies of different duocarmycin based glycosidic prodrugs for their use in the antibody-directed enzyme prodrug therapy   [0296] 
Asymmetric synthesis and biological evaluation of glycosidic prodrugs for a selective cancer therapy   [0296] 
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Enantio- and diastereoselective synthesis of duocarmycine-based prodrugs for a selective treatment of cancer by epoxide opening   [0296] 
Selective treatment of cancer: synthesis, biological evaluation and structural elucidation of novel analogues of the antibiotic CC-1065 and the duocarmycins   [0296] 
Antitumor agents: development of highly potent glycosidic duocarmycin analogues for selective cancer therapy   [0296] 
Investigation of reactivity and selectivity of DNA-alkylating duocarmycin analogues by high-resolution mass spectrometry   [0296] 
Enzyme and proton-activated prodrugs for a selective cancer therapy   [0296] 
Proof of principle in the selective treatment of cancer by antibody-directed enzyme prodrug therapy: the development of a highly potent prodrug   [0296] 
Highly selective glycosylated prodrugs of cytostatic CC-1065 analogues for antibody-directed enzyme tumor therapy   [0296] 
A strategy for tumor-selective chemotherapy by enzymatic liberation of seco-duocarmycin SA-derivatives from nontoxic prodrugs   [0296] 
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Synthesis, biological evaluation, and live cell imaging of novel fluorescent duocarmycin analogs   [0296] 
Synthesis of Fluorescence-Labelled Glycosidic Prodrugs Based on the Cytotoxic Antibiotic Duocarmycin   [0296] 
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Prodrugs of the Cytostatic CC-1065 That Can Be Activated in a Tumor-Selective Manner   [0296] 
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