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Es wird ein Verfahren zur Herstellung von Imidazopyridinderivaten der allgemeinen Formel beschrieben.Dabei wird ein 2-Amino-3-nitropyridin in Gegenwart eines Hydrierkatalysators hydriert und das Hydrierprodukt mit einer gleichzeitig im Reaktionsgemisch vorliegenden Carbonsäure zum Endprodukt kondensiert.Die Imidazopyridinderivate sind Zwischenprodukte für die Herstellung von Angiotensin-II-Antagonisten.
Es wird ein Verfahren zur Herstellung von Imidazopyridinderivaten der allgemeinen Formel beschrieben.Dabei wird ein 2-Amino-3-nitropyridin in Gegenwart eines Hydrierkatalysators hydriert und das Hydrierprodukt mit einer gleichzeitig im Reaktionsgemisch vorliegenden Carbonsäure zum Endprodukt kondensiert.Die Imidazopyridinderivate sind Zwischenprodukte für die Herstellung von Angiotensin-II-Antagonisten.
de
European Patent Office
EP0656358
EP 0656358
C07D 471/04
C07D471/04
C07D235/00
C07D221/00
Process for the preparation of imidazopyridinderivatives
Verfahren zur Herstellung von Imidazopyridinderivaten - European Patent Office - EP 0656358 A1
Verfahren zur Herstellung von Imidazopyridinderivaten - European Patent Office - EP 0656358 A1
Adobe PDF Library 8.0
"EP0656358"; "EP 0656358"; "C07D 471/04"; "C07D471/04"; "C07D235/00"; "C07D221/00"; "Process for the preparation of imidazopyridinderivatives"
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1993-12-01
C07D 471/04
C07D471/04
C07D235/00
C07D221/00
LONZA AG
Kuo, David L. Dr.
Eyer, Martin, Dr.
Roduit, Jean-Paul, Dr.
Wellig, Alain
Weinhold, Peter, Dr.
Verfahren zur Herstellung von Imidazopyridinderivaten
Verfahren zur Herstellung von Imidazopyridinderivaten
Process for the preparation of imidazopyridinderivatives
Procédé pour la préparation de dérivés d'imidazopyridine
Es wird ein Verfahren zur Herstellung von Imidazopyridinderivaten der allgemeinen Formel beschrieben.Dabei wird ein 2-Amino-3-nitropyridin in Gegenwart eines Hydrierkatalysators hydriert und das Hydrierprodukt mit einer gleichzeitig im Reaktionsgemisch vorliegenden Carbonsäure zum Endprodukt kondensiert.Die Imidazopyridinderivate sind Zwischenprodukte für die Herstellung von Angiotensin-II-Antagonisten.
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