| (19) |
 |
|
(11) |
EP 0 187 390 A3 |
| (12) |
EUROPEAN PATENT APPLICATION |
| (88) |
Date of publication A3: |
|
25.03.1987 Bulletin 1987/13 |
| (43) |
Date of publication A2: |
|
16.07.1986 Bulletin 1986/29 |
| (22) |
Date of filing: 30.12.1985 |
|
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| (84) |
Designated Contracting States: |
|
AT BE CH DE FR GB IT LI LU NL SE |
| (30) |
Priority: |
31.12.1984 US 687628
|
| (71) |
Applicant: MERRELL DOW PHARMACEUTICALS INC. |
|
() |
|
| (72) |
Inventors: |
|
- Bargar, Thomas M.
()
- Broersma, Robert, Jr.
()
- McCarthy, James R.
()
|
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| |
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| (54) |
Novel allylic amines |
(57) 57 This invention relates to novel β-methylene- thiophenethanamines which are mechanism-based
inhibitors of dopamine beta-hydroxylase useful as antihypertensive agents.