(19)
(11) EP 2 831 070 A1

(12)

(43) Date of publication:
04.02.2015 Bulletin 2015/06

(21) Application number: 13768214.2

(22) Date of filing: 21.03.2013
(51) International Patent Classification (IPC): 
C07D 453/02(2006.01)
A61K 31/439(2006.01)
C07D 401/12(2006.01)
A61P 13/00(2006.01)
(86) International application number:
PCT/KR2013/002358
(87) International publication number:
WO 2013/147458 (03.10.2013 Gazette 2013/40)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(30) Priority: 28.03.2012 KR 20120031492

(71) Applicant: Kyung Dong Pharm. Co., Ltd.
Yanggam-myeon, Hwaseong-si, Gyeonggi-do 445-931 (KR)

(72) Inventors:
  • LEE, Byoung Suk
    Seoul 137-755 (KR)
  • SHIN, Sang Hoon
    Suwon-si Gyeonggi-do 440-320 (KR)
  • LEE, Ki Young
    Osan-si Gyeonggi-do 447-747 (KR)

(74) Representative: McConchie, Connor Fraser 
D Young & Co LLP 120 Holborn
London EC1N 2DY
London EC1N 2DY (GB)

   


(54) PROCESS OF PREPARING SOLIFENACIN OR SALT THEREOF, AND NOVEL INTERMEDIATE USED IN THE PROCESS