(19)
(11) EP 0 097 013 A3

(12) EUROPEAN PATENT APPLICATION

(88) Date of publication A3:
02.01.1985 Bulletin 1985/01

(43) Date of publication A2:
28.12.1983 Bulletin 1983/52

(21) Application number: 83303256

(22) Date of filing: 06.06.1983
(84) Designated Contracting States:
BE CH DE FR GB IT LI LU NL SE

(30) Priority: 07.06.1982 US 385602
07.03.1983 US 472439

(71) Applicant: ELI LILLY AND COMPANY
 ()

(72) Inventors:
  • Krumkalns, Eriks Victor
     ()
  • Smiley, David Lee
     ()

   


(54) Fungicidal heterocyclic amines


(57) eterocyclic amines of the formula (I):

or an agronomically acceptable acid addition or quaternary ammonium salt thereof wherein

R' is pyridyl, pyrimidinyl, pyrazinyl, pyridazinyl, or one of said groups substituted with one or two groups independently selected from halogen, C,-C4 alkyl, C,-C4 haloalkyl, and C1-C4 haloalkoxy; q is 0, or 2;

R2, if applicable, is hydrogen, C1-C4 alkyl, or a group of the formula (II):

wherein R3 and R4 are independently selected from hydrogen, C1-C6 alkyl, C1-C6 alkoxy, C3-C8 cycloalkyl, C1-C6 alkylthio, halogen, C1-C6 haloalkyl, C1-C6 haloalkoxy, nitro, and cyano; and r is 0 or 1;

R5 is C1-C10 alkyl, C2-C10 alkenyl, C1-C10 alkoxy, C1-C10 haloalkyl, C1-C10 haloalkoxy, C3-C8 cycloalkyl, 1,3-benzodioxyl, or a group of the formula (III):

wherein:

s is 0,1,2 or 3

R6 is independently hydrogen or C1-C4 alkyl; and

R7 and R8 are independently selected from hydrogen, C1-C6 alkyl, C1-C6 alkoxy, C3-C8 cycloalkyl, C1-C6 alkylthio, halogen, C1-C6 haloalkyl, C1-C6 haloalkoxy, nitro, cyano, or a group of the formula (IV)

wherein:

Z is oxygen, sulfur, -(CH2)t-, or a direct link, t being 0,1,2, or 3, and

R9 and R10 are independently selected from hydrogen, C1-C6 alkyl, C1-C6 alkoxy, C3-C8 cycloalkyl, C1-C6 alkylthio, halogen, C1-C6 haloalkyl, C,-C6 haloalkoxy, nitro and cyano;

R", R'3 and, if applicable, R12 are independently hydrogen or C1-C4 alkyl;

m is 0 or 1;and

X is sulfur or oxygen,

are useful as plant fungicides and aquatic plant growth regulators.







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