(19)
(11) EP 0 247 033 A1

(12)

(43) Date of publication:
02.12.1987 Bulletin 1987/49

(21) Application number: 85905687.0

(22) Date of filing: 25.10.1985
(51) International Patent Classification (IPC): 
C07K 7/ 16( . )
 A61K 38/ 00( . )
(86) International application number:
PCT/US1985/002104
(87) International publication number:
WO 1987/002676 (07.05.1987 Gazette 1987/10)
(84) Designated Contracting States:
AT BE CH DE FR GB IT LI LU NL SE

(71) Applicant: GIBSON-STEPHENS NEUROPHARMACEUTICALS, INC.
Tucson, AZ 85719 (US)

(72) Inventors:
  • HRUBY, Victor, J.
    Tucson, AZ 85716 (US)
  • ROCKWAY, Todd, W.
    San Diego, CA 92107 (US)

   


(54) CONFORMATIONALLY CONSTRAINED OXYTOCIN ANTAGONISTS WITH PROLONGED BIOLOGICAL ACTIVITIES