(19)
(11) EP 0 293 432 A1

(12)

(43) Date of publication:
07.12.1988 Bulletin 1988/49

(21) Application number: 88900014.0

(22) Date of filing: 30.10.1987
(51) International Patent Classification (IPC): 
A61K 31/ 00( . )
A61K 31/ 34( . )
A61K 31/ 405( . )
A61K 31/ 47( . )
A61K 31/ 575( . )
A61P 43/ 00( . )
C07C 53/ 128( . )
C07C 59/ 64( . )
C07C 63/ 06( . )
C07C 63/ 70( . )
C07C 67/ 00( . )
C07C 227/ 00( . )
C07C 231/ 00( . )
C07C 237/ 12( . )
C07K 14/ 81( . )
A61K 31/ 19( . )
A61K 31/ 40( . )
A61K 31/ 445( . )
A61K 31/ 50( . )
A61K 38/ 00( . )
C07C 51/ 00( . )
C07C 57/ 30( . )
C07C 59/ 84( . )
C07C 63/ 36( . )
C07C 65/ 21( . )
C07C 201/ 00( . )
C07C 229/ 42( . )
C07C 233/ 54( . )
C07K 5/ 06( . )
(86) International application number:
PCT/EP1987/000664
(87) International publication number:
WO 1988/003020 (05.05.1988 Gazette 1988/10)
(84) Designated Contracting States:
AT BE CH DE FR GB IT LI LU NL SE

(30) Priority: 31.10.1986 NL 19860002767

(71) Applicant: NV GANTAX PHARMACEUTICA
B-2520 Edegem (BE)

(72) Inventors:
  • JANSEN, Frans, Herwig, Jan
    B-2360 Oud Turnhout (BE)
  • DE COCK, Etienne, Jacquy
    B-1820 Grimbergen (BE)

(74) Representative: van 't Holt, Henk 
Patent Attorney/Octrooigemachtigde Churchilllaan 30
NL-5224 BV 's-Hertogenbosch
NL-5224 BV 's-Hertogenbosch (NL)

   


(54) ORGANIC ACID ANHYDRIDE AND PHARMACEUTICAL COMPOSITION ON A PRODRUG BASE