(19)
(11) EP 0 328 203 A3

(12) EUROPEAN PATENT APPLICATION

(88) Date of publication A3:
14.03.1990 Bulletin 1990/11

(43) Date of publication A2:
16.08.1989 Bulletin 1989/33

(21) Application number: 89200253.6

(22) Date of filing: 06.02.1989
(51) International Patent Classification (IPC)4: C07D 403/06, C07D 409/14
(84) Designated Contracting States:
AT BE CH DE ES FR GB GR IT LI LU NL SE

(30) Priority: 12.02.1988 US 155464

(71) Applicant: JANSSEN PHARMACEUTICA N.V.
B-2340 Beerse (BE)

(72) Inventors:
  • Raeymaekers, Alfons H.M.
    B-2340-Beerse (BE)
  • Freyne, Eddy J.E.
    B-2638-Rumst (BE)


(56) References cited: : 
   
       


    (54) [5(6) (1H-azole-1-ylmethyl)benzimidazole] carbamates


    (57) Novel [5(6) (1H-azole-1-ylmethyl)benzimidazole]carbamates having the formula

    wherein
    R is C₁-₆alkyl, C₃₋₆cycloalkyl, thienyl or substituted phenyl;
    R¹ is C₁₋₆alkyl;
    R² is hydrogen or C₁₋₆alkyl;
    Q is N or CH;
    pharmaceutical compositions containing said compounds as active ingredient; methods of preparing said compounds and compositions.





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