TRI- AND TETRA-SUBSTITUTED-OXETANES AND TETRAHYDROFURANS AND INTERMEDIATES THEREOF - Patent 0386143

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EP 0 386 143 A1

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(43)	Date of publication:
	12.09.1990 Bulletin 1990/37

(21)	Application number: 89900481.0

(22)	Date of filing: 18.11.1988

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International Patent Classification (IPC):

C07D 473/ 08^{( . )}
A61K 31/ 415^{( . )}
A61K 31/ 44^{( . )}
A61K 31/ 4433^{( . )}
A61K 31/ 52^{( . )}
A61P 29/ 00^{( . )}
A61P 37/ 08^{( . )}
C07D 405/ 14^{( . )}
C07D 417/ 14^{( . )}
C07D 493/ 08^{( . )}

A61K 31/ 41^{( . )}
A61K 31/ 425^{( . )}
A61K 31/ 443^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 522^{( . )}
A61P 31/ 00^{( . )}
C07D 405/ 06^{( . )}
C07D 409/ 14^{( . )}
C07D 473/ 10^{( . )}
C07D 521/ 00^{( . )}

(86)	International application number:
	PCT/US1988/003987

(87)	International publication number:
	WO 1989/004829 (01.06.1989 Gazette 1989/12)

(84)	Designated Contracting States:
	AT BE CH DE FR GB IT LI LU NL SE

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Priority:

20.11.1987 US 19870123500

(71)	Applicant: SCHERING CORPORATION
	Kenilworth New Jersey 07033 (US)

(72)	Inventors:
	SAKSENA, Anil, K. Upper Montclair, NJ 07043 (US) GIRIJAVALLABHAN, Viyyoor, M. Parsippany, NJ 07054 (US) GANGULY, Ashit, K. Upper Montclair, NJ 07043 (US) RANE, Dinanath, F. Morganville, NJ 07751 (US)

(74)	Representative: Ritter, Stephen David, et al
	Mathys & Squire 100 Grays Inn Road London WC1X 8AL London WC1X 8AL (GB)

(54)	TRI- AND TETRA-SUBSTITUTED-OXETANES AND TETRAHYDROFURANS AND INTERMEDIATES THEREOF