(19)
(11) EP 0 397 779 A1

(12)

(43) Date of publication:
22.11.1990 Bulletin 1990/47

(21) Application number: 89902438.0

(22) Date of filing: 27.01.1989
(51) International Patent Classification (IPC): 
C07D 263/ 06( . )
A61P 9/ 12( . )
C07D 493/ 08( . )
C07K 5/ 02( . )
C07K 5/ 10( . )
C07K 14/ 81( . )
A61K 38/ 55( . )
C07C 271/ 48( . )
C07F 7/ 18( . )
C07K 5/ 08( . )
C07K 9/ 00( . )
(86) International application number:
PCT/US1989/000247
(87) International publication number:
WO 1989/007109 (10.08.1989 Gazette 1989/18)
(84) Designated Contracting States:
AT BE CH DE FR GB IT LI LU NL SE

(30) Priority: 01.02.1988 US 19880151129

(71) Applicant: THE UPJOHN COMPANY
Kalamazoo, MI 49001 (US)

(72) Inventors:
  • BUNDY, Gordon, L.
    Portage, MI 49002 (US)
  • THAISRIVONGS, Suvit
    Portage, MI 49002 (US)
  • NELSON, Norman, A.
    Galesburg, MI 49053 (US)
  • HESTER, Jackson, B., Jr.
    Galesburg, MI 49053 (US)
  • FISHER, Jed, F.
    Three Rivers, MI 49093 (US)
  • LIPTON, Michael, F.
    Kalamazoo, MI 49001 (US)

(74) Representative: Perry, Robert Edward, et al 
GILL JENNINGS & EVERY Broadgate House 7 Eldon Street
London EC2M 7LH
London EC2M 7LH (GB)

   


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