NOVEL RENIN-INHIBITING PEPTIDES HAVING A DIHYDROXYETHYLENE ISOSTERE TRANSITION STATE INSERT - Patent 0406228

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EP 0 406 228 A1

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(43)	Date of publication:
	09.01.1991 Bulletin 1991/02

(21)	Application number: 87901865.0

(22)	Date of filing: 13.02.1987

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International Patent Classification (IPC):

C07D 233/ 54^{( . )}

C07K 5/ 02^{( . )}

(86)	International application number:
	PCT/US1987/000291

(87)	International publication number:
	WO 1987/005302 (11.09.1987 Gazette 1987/20)

(84)	Designated Contracting States:
	BE CH DE FR GB IT LI LU NL SE

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Priority:

27.02.1986 US 19860833993
05.09.1986 US 19860904149

(71)	Applicant: THE UPJOHN COMPANY
	Kalamazoo, Michigan 49001 (US)

(72)	Inventor:
	THAISRIVONGS, Suvit Portage, MI 49002 (US)

(74)	Representative: Perry, Robert Edward, et al
	GILL JENNINGS & EVERY Broadgate House 7 Eldon Street London EC2M 7LH London EC2M 7LH (GB)

(54)	NOVEL RENIN-INHIBITING PEPTIDES HAVING A DIHYDROXYETHYLENE ISOSTERE TRANSITION STATE INSERT